SCHEMBL19795461

SCHEMBL19795461

Cc1ccc(N(c2ccc(C=C(c3ccccc3)c3ccccc3)cc2)c2ccc(C)cc2C)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 6/20 0.49
CYP19A1 P11511 1/20 0.40
CYP11B2 P19099 1/20 0.40
ESR1 P03372 1/20 0.37
TRPM8 Q7Z2W7 1/20 0.37
MAPT P10636 5/20 0.36
ALDH1A1 P00352 3/20 0.36
CYP3A4 P08684 1/20 0.36
HPGD P15428 1/20 0.36
RAB9A P51151 2/20 0.36
MAPK1 P28482 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
LMNA P02545 2/20 0.36
KMT2A Q03164 2/20 0.36
NPSR1 Q6W5P4 2/20 0.36
CYP2D6 P10635 1/20 0.36
MEN1 O00255 1/20 0.36
CRHBP P24387 1/20 0.36
CRHR2 Q13324 1/20 0.36
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12576285 0.99 PTGS2 (0.51) PTGS2CYP19A1CYP11B2ESR1TRPM8
SCHEMBL13050002 0.99 PTGS2 (0.51) PTGS2CYP19A1CYP11B2ESR1TRPM8
SCHEMBL14769858 0.99 PTGS2 (0.51) PTGS2CYP19A1CYP11B2ESR1TRPM8
SCHEMBL10057475 0.99 PTGS2 (0.47) PTGS2CYP19A1CYP11B2ESR1MAPT
SCHEMBL13679109 0.95 PTGS2 (0.44) PTGS2CYP19A1CYP11B2ESR1TRPM8
SCHEMBL15478868 0.95 PTGS2 (0.44) PTGS2CYP19A1CYP11B2ESR1TRPM8
SCHEMBL12576286 0.93 PTGS2 (0.47) PTGS2ESR1MAPTALDH1A1CYP3A4
SCHEMBL21029949 0.93 PTGS2 (0.47) PTGS2ESR1MAPTALDH1A1CYP3A4
SCHEMBL25053712 0.91 PTGS2 (0.41) PTGS2CYP19A1CYP11B2ESR1TRPM8
SCHEMBL2614959 0.91 PTGS2 (0.44) PTGS2CYP19A1CYP11B2ESR1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230259046-A1 ELECTROPHOTOGRAPHIC PHOTORECEPTOR, CARTRIDGE USING SAME, AND IMAGE FORMING DEVICE MITSUBISHI CHEMICAL CORPORATION (JP) 2023-08-17 US disclosed
US-20230259046-A1 ELECTROPHOTOGRAPHIC PHOTORECEPTOR, CARTRIDGE USING SAME, AND IMAGE FORMING DEVICE MITSUBISHI CHEMICAL CORPORATION (JP) 2023-08-17 US disclosed
US-11169453-B2 Electrophotographic photosensitive member, process cartridge and electrophotographic apparatus CANON KABUSHIKI KAISHA (JP) 2021-11-09 US disclosed
US-20200393772-A1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE AND ELECTROPHOTOGRAPHIC APPARATUS CANON KABUSHIKI KAISHA (JP) 2020-12-17 US disclosed
US-10324386-B2 Electrophotographic photoreceptor, image forming apparatus, image forming method, production method of electrophotographic photoreceptor Konica Minolta, Inc. (JP) 2019-06-18 US disclosed
US-10203615-B2 Electrophotographic photoreceptor, image forming apparatus, image forming method, and method of producing electrophotographic photoreceptor Konica Minolta, Inc. (JP) 2019-02-12 US disclosed
US-20180224761-A1 ELECTROPHOTOGRAPHIC PHOTORECEPTOR, IMAGE FORMING APPARATUS, IMAGE FORMING METHOD, PRODUCTION METHOD OF ELECTROPHOTOGRAPHIC PHOTORECEPTOR Konica Minolta, Inc. (JP) 2018-08-09 US disclosed
US-20180224761-A1 ELECTROPHOTOGRAPHIC PHOTORECEPTOR, IMAGE FORMING APPARATUS, IMAGE FORMING METHOD, PRODUCTION METHOD OF ELECTROPHOTOGRAPHIC PHOTORECEPTOR Konica Minolta, Inc. (JP) 2018-08-09 US disclosed
US-20180173120-A1 ELECTROPHOTOGRAPHIC PHOTORECEPTOR, IMAGE FORMING APPARATUS, IMAGE FORMING METHOD, AND METHOD OF PRODUCING ELECTROPHOTOGRAPHIC PHOTORECEPTOR Konica Minolta, Inc. (JP) 2018-06-21 US disclosed
US-20180173120-A1 ELECTROPHOTOGRAPHIC PHOTORECEPTOR, IMAGE FORMING APPARATUS, IMAGE FORMING METHOD, AND METHOD OF PRODUCING ELECTROPHOTOGRAPHIC PHOTORECEPTOR Konica Minolta, Inc. (JP) 2018-06-21 US disclosed
US-20180024450-A1 ELECTROPHOTOGRAPHIC PHOTORECEPTOR, METHOD OF PRODUCING ELECTROPHOTOGRAPHIC PHOTORECEPTOR, AND APPARATUS OF FORMING ELECTROPHOTOGRAPHIC IMAGE Konica Minolta, Inc. (JP) 2018-01-25 US disclosed
US-20180024450-A1 ELECTROPHOTOGRAPHIC PHOTORECEPTOR, METHOD OF PRODUCING ELECTROPHOTOGRAPHIC PHOTORECEPTOR, AND APPARATUS OF FORMING ELECTROPHOTOGRAPHIC IMAGE Konica Minolta, Inc. (JP) 2018-01-25 US disclosed