SCHEMBL19795462

SCHEMBL19795462

C/C(=C\c1ccc(N(c2ccccc2)c2ccccc2)cc1)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.50
ESR2 Q92731 1/20 0.50
PTGS2 P35354 5/20 0.47
PTGS1 P23219 4/20 0.47
ALDH1A1 P00352 7/20 0.46
MAPT P10636 6/20 0.46
KMT2A Q03164 5/20 0.46
LMNA P02545 2/20 0.46
GAA P10253 1/20 0.46
L3MBTL1 Q9Y468 2/20 0.45
RAB9A P51151 2/20 0.45
MAPK1 P28482 2/20 0.45
NQO2 P16083 3/20 0.42
MEN1 O00255 3/20 0.41
KDM4E B2RXH2 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10746258 1.00 ESR1 (0.50) ESR1ESR2PTGS2PTGS1ALDH1A1
SCHEMBL4585196 0.98 ESR1 (0.52) ESR1ESR2PTGS2PTGS1ALDH1A1
SCHEMBL13808874 0.93 ESR1 (0.47) ESR1ESR2PTGS2PTGS1ALDH1A1
SCHEMBL11060353 0.93 ESR1 (0.50) ESR1ESR2PTGS2PTGS1ALDH1A1
SCHEMBL14199384 0.91 ESR1 (0.46) ESR1ESR2PTGS2PTGS1ALDH1A1
SCHEMBL4585187 0.91 ESR1 (0.52) ESR1ESR2PTGS2PTGS1ALDH1A1
SCHEMBL13807875 0.86 ESR1 (0.45) ESR1ESR2PTGS2PTGS1ALDH1A1
SCHEMBL25909565 0.85 PTGS1 (0.65) ESR1ESR2PTGS2PTGS1ALDH1A1
SCHEMBL14570726 0.85 PTGS1 (0.65) ESR1ESR2PTGS2PTGS1ALDH1A1
SCHEMBL14077323 0.82 RELA (0.41) PTGS2PTGS1ALDH1A1MAPTNQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11169453-B2 Electrophotographic photosensitive member, process cartridge and electrophotographic apparatus CANON KABUSHIKI KAISHA (JP) 2021-11-09 US disclosed
US-20200393772-A1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE AND ELECTROPHOTOGRAPHIC APPARATUS CANON KABUSHIKI KAISHA (JP) 2020-12-17 US disclosed
US-10324386-B2 Electrophotographic photoreceptor, image forming apparatus, image forming method, production method of electrophotographic photoreceptor Konica Minolta, Inc. (JP) 2019-06-18 US disclosed
US-10203615-B2 Electrophotographic photoreceptor, image forming apparatus, image forming method, and method of producing electrophotographic photoreceptor Konica Minolta, Inc. (JP) 2019-02-12 US disclosed
US-20180224761-A1 ELECTROPHOTOGRAPHIC PHOTORECEPTOR, IMAGE FORMING APPARATUS, IMAGE FORMING METHOD, PRODUCTION METHOD OF ELECTROPHOTOGRAPHIC PHOTORECEPTOR Konica Minolta, Inc. (JP) 2018-08-09 US disclosed
US-20180224761-A1 ELECTROPHOTOGRAPHIC PHOTORECEPTOR, IMAGE FORMING APPARATUS, IMAGE FORMING METHOD, PRODUCTION METHOD OF ELECTROPHOTOGRAPHIC PHOTORECEPTOR Konica Minolta, Inc. (JP) 2018-08-09 US disclosed
US-20180173120-A1 ELECTROPHOTOGRAPHIC PHOTORECEPTOR, IMAGE FORMING APPARATUS, IMAGE FORMING METHOD, AND METHOD OF PRODUCING ELECTROPHOTOGRAPHIC PHOTORECEPTOR Konica Minolta, Inc. (JP) 2018-06-21 US disclosed
US-20180173120-A1 ELECTROPHOTOGRAPHIC PHOTORECEPTOR, IMAGE FORMING APPARATUS, IMAGE FORMING METHOD, AND METHOD OF PRODUCING ELECTROPHOTOGRAPHIC PHOTORECEPTOR Konica Minolta, Inc. (JP) 2018-06-21 US disclosed
US-20180024450-A1 ELECTROPHOTOGRAPHIC PHOTORECEPTOR, METHOD OF PRODUCING ELECTROPHOTOGRAPHIC PHOTORECEPTOR, AND APPARATUS OF FORMING ELECTROPHOTOGRAPHIC IMAGE Konica Minolta, Inc. (JP) 2018-01-25 US disclosed
US-20180024450-A1 ELECTROPHOTOGRAPHIC PHOTORECEPTOR, METHOD OF PRODUCING ELECTROPHOTOGRAPHIC PHOTORECEPTOR, AND APPARATUS OF FORMING ELECTROPHOTOGRAPHIC IMAGE Konica Minolta, Inc. (JP) 2018-01-25 US disclosed