SCHEMBL1979661

SCHEMBL1979661

CC(C)(C)OC(=O)NCC1(Cn2c(C(=O)O)cc3ccc(C(=O)O)cc32)CC1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.38
CCR9 P51686 10/20 0.37
P2RY14 Q15391 1/20 0.35
HCRTR2 O43614 1/20 0.35
ACACB O00763 1/20 0.34
ACACA Q13085 1/20 0.34
CNR2 P34972 1/20 0.33
MAPT P10636 1/20 0.33
NPFFR1 Q9GZQ6 1/20 0.33
NPFFR2 Q9Y5X5 1/20 0.33
GPR35 Q9HC97 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1979671 0.96 BRD4 (0.37) BRD4CCR9P2RY14HCRTR2ACACB
SCHEMBL1977977 0.85 MEN1 (0.39) BRD4MAPT
SCHEMBL14904443 0.84 MEN1 (0.38) BRD4HCRTR2
SCHEMBL12598985 0.82 MEN1 (0.38) BRD4MAPT
SCHEMBL14904448 0.81 MEN1 (0.37) BRD4CNR2
SCHEMBL1983809 0.80 ALDH1A1 (0.37) BRD4HCRTR2MAPT
SCHEMBL1978852 0.79 ATM (0.39) MAPT
SCHEMBL14904457 0.79 MEN1 (0.36) CNR2MAPT
SCHEMBL12598785 0.73 BRD4 (0.42) BRD4CNR2MAPT
SCHEMBL6207500 0.71 TSHR (0.42) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2509980-A1 HETEROCYCLIC COMPOUNDS CONTAINING AN INDOLE CORE Boehringer Ingelheim International GmbH (DE) 2012-10-17 EP disclosed
WO-2011071716-A1 HETEROCYCLIC COMPOUNDS CONTAINING AN INDOLE CORE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-06-16 WO disclosed