SCHEMBL1980252

SCHEMBL1980252

Nc1ncnc2c1ncn2[C@@]1(O)[C@H](O)CO[C@@H]1CO

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 4/20 0.52
ADORA2A P29274 3/20 0.52
SLC28A1 O00337 3/20 0.52
GMPS P49915 1/20 0.49
PI4KA P42356 3/20 0.46
PI4K2B Q8TCG2 3/20 0.46
PI4K2A Q9BTU6 3/20 0.46
PI4KB Q9UBF8 3/20 0.46
AHCY P23526 4/20 0.46
EGFR P00533 1/20 0.44
ERBB2 P04626 1/20 0.44
ADORA2B P29275 2/20 0.44
SLC28A2 O43868 2/20 0.44
DPP4 P27487 1/20 0.44
MEN1 O00255 1/20 0.44
MAP3K7 O43318 1/20 0.44
GAPDH P04406 1/20 0.44
MAPK1 P28482 1/20 0.44
ADORA1 P30542 1/20 0.44
STAT6 P42226 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8590840 1.00 ADORA3 (0.52) ADORA3ADORA2ASLC28A1GMPSPI4KA
SCHEMBL5607133 0.84 ADORA2A (0.36) ADORA3ADORA2ASLC28A1GMPSAHCY
SCHEMBL15741480 0.83 AHCY (0.47) ADORA3ADORA2ASLC28A1AHCYADORA2B
SCHEMBL27214952 0.80 AHCY (0.35) ADORA3ADORA2ASLC28A1AHCYADORA1
SCHEMBL1934830 0.79 ADORA2A (0.51) ADORA3ADORA2ASLC28A1GMPSPI4KA
SCHEMBL10785491 0.78 ADORA3 (0.31) ADORA3ADORA2ASLC28A1
SCHEMBL23025515 0.78 ADORA3 (0.53) ADORA3ADORA2ASLC28A1GMPSPI4KA
SCHEMBL25521510 0.78 ADORA3 (0.53) ADORA3ADORA2ASLC28A1GMPSPI4KA
SCHEMBL9667894 0.77 ADORA3 (0.46) ADORA3MEN1KMT2ASMN1; SMN2
SCHEMBL9450389 0.76 HSP90AA1 (0.36) ADORA3ADORA2ASLC28A1AHCYADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992010198-A1 IMMUNOTHERAPEUTIC AGENTS, COMPOSITIONS AND METHODS JOHNSON & JOHNSON RESEARCH PTY LIMITED (AU) 1992-06-25 WO claimed
EP-0121635-A1 3',5',-Diarabinosides, their preparation and their therapeutical application SYNTHELABO (FR) 1984-10-17 EP claimed
EP-2509990-A1 NOVEL PHOSPH(ON)ATE- AND SULF(ON)ATE-BASED PHOSPHATE MODIFIED NUCLEOSIDES USEFUL AS SUBSTRATES FOR POLYMERASES AND AS ANTIVIRAL AGENTS Katholieke Universiteit Leuven, K.U. Leuven R&D (BE) 2012-10-17 EP disclosed
US-20120245029-A1 NOVEL PHOSPH(ON)ATE- AND SULF(ON)ATE-BASED PHOSPHATE MODIFIED NUCLEOSIDES USEFUL AS SUBSTRATES FOR POLYMERASES AND AS ANTIVIRAL AGENTS KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2012-09-27 US disclosed
WO-2011069688-A1 NOVEL PHOSPH(ON)ATE- AND SULF(ON)ATE-BASED PHOSPHATE MODIFIED NUCLEOSIDES USEFUL AS SUBSTRATES FOR POLYMERASES AND AS ANTIVIRAL AGENTS KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2011-06-16 WO disclosed
EP-0891374-A4 UNIQUE ASSOCIATED KAPOSI'S SARCOMA VIRUS SEQUENCES AND USES THEREOF UNIV COLUMBIA (US) 1999-04-07 EP disclosed
EP-0891374-A1 UNIQUE ASSOCIATED KAPOSI'S SARCOMA VIRUS SEQUENCES AND USES THEREOF The Trustees of Columbia University in the City of New York (US) 1999-01-20 EP disclosed
WO-1997027208-A1 UNIQUE ASSOCIATED KAPOSI'S SARCOMA VIRUS SEQUENCES AND USES THEREOF THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 1997-07-31 WO disclosed
EP-0674529-A1 LIPID PRODRUGS FOR ORAL ADMINISTRATION NeXstar Pharmaceuticals, Inc. (US) 1995-10-04 EP disclosed
WO-1994013324-A1 LIPID PRODRUGS FOR ORAL ADMINISTRATION VESTAR, INC. (US) 1994-06-23 WO disclosed
EP-0517859-A1 OLIGONUCLEOTIDE THERAPIES FOR MODULATING THE EFFECTS OF HERPESVIRUSES ISIS PHARMACEUTICALS, INC. (US) 1992-12-16 EP disclosed
WO-1991012811-A1 OLIGONUCLEOTIDE THERAPIES FOR MODULATING THE EFFECTS OF HERPESVIRUSES ISIS PHARMACEUTICALS, INC. (US) 1991-09-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120245029-A1 NOVEL PHOSPH(ON)ATE- AND SULF(ON)ATE-BASED PHOSPHATE MODIFIED NUCLEOSIDES USEFUL AS SUBSTRATES FOR POLYMERASES AND AS ANTIVIRAL AGENTS TYMP, PNP, MTAP ADORA3 100/4885ADORA2A 191/4885SLC28A1 386/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.