SCHEMBL1982960

SCHEMBL1982960

OC1COc2cc(F)ccc2C1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.41
ESR2 Q92731 1/20 0.41
TTR P02766 1/20 0.41
RIPK1 Q13546 1/20 0.37
AKR1B1 P15121 1/20 0.37
CYP19A1 P11511 1/20 0.35
CA2 P00918 1/20 0.35
HIF1A Q16665 1/20 0.34
ACHE P22303 1/20 0.34
ALOX15B O15296 1/20 0.34
ALOX15 P16050 1/20 0.34
ALOX12 P18054 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
MAOB P27338 3/20 0.33
HTR1A P08908 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31031129 0.80 ESR1 (0.63) ESR1ESR2TTRCA2ALOX15B
SCHEMBL18983645 0.80 ESR1 (0.63) ESR1ESR2TTRCA2ALOX15B
SCHEMBL25082619 0.79 ACHE (0.41) ESR1ESR2TTRRIPK1AKR1B1
SCHEMBL8354476 0.79 ACHE (0.41) ESR1ESR2TTRRIPK1AKR1B1
SCHEMBL13977477 0.79 MAP3K14 (0.44) ESR1ESR2TTRCYP19A1CA2
SCHEMBL24214986 0.78 LTB4R (0.40) ESR1ESR2TTRRIPK1AKR1B1
SCHEMBL30292064 0.77 HDAC1 (0.44) ESR1ESR2RIPK1AKR1B1HDAC1
SCHEMBL22165402 0.77 HDAC1 (0.44) ESR1ESR2RIPK1AKR1B1HDAC1
SCHEMBL27883209 0.77 HDAC1 (0.44) ESR1ESR2RIPK1AKR1B1HDAC1
SCHEMBL23558482 0.75 LTB4R (0.40) ESR1ESR2TTRHDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2509950-A1 5-AMINO- 4-HYDROXYPENTOYL AMIDES Janssen R&D Ireland (IE) 2012-10-17 EP disclosed
WO-2011070131-A1 5-AMINO- 4-HYDROXYPENTOYL AMIDES TIBOTEC PHARMACEUTICALS (IE) 2011-06-16 WO disclosed