SCHEMBL19831386

SCHEMBL19831386

C=C(C)[C@H](NS(=O)(=O)c1ccc(F)cc1)C(=O)N[C@H](C=O)CC(C)C

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 7/20 0.48
CTSB P07858 2/20 0.42
CTSL P07711 1/20 0.42
CTSS P25774 1/20 0.42
CTSK P43235 1/20 0.42
MMP1 P03956 2/20 0.40
MMP2 P08253 2/20 0.40
MMP3 P08254 2/20 0.40
MMP7 P09237 2/20 0.40
MMP9 P14780 2/20 0.40
MMP13 P45452 2/20 0.40
GFER P55789 1/20 0.39
MMP8 P22894 1/20 0.37
MMP14 P50281 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
GAA P10253 1/20 0.37
SLC1A3 P43003 1/20 0.37
SLC1A2 P43004 1/20 0.37
SLC1A1 P43005 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6026500 0.83 CAPN1 (0.66) CAPN1CTSBCTSLCTSSCTSK
SCHEMBL3913553 0.83 CAPN1 (0.66) CAPN1CTSBCTSLCTSSCTSK
SCHEMBL3904669 0.83 CAPN1 (0.66) CAPN1CTSBCTSLCTSSCTSK
SCHEMBL5363846 0.83 CAPN1 (0.66) CAPN1CTSBCTSLCTSSCTSK
SCHEMBL1907361 0.83 CAPN1 (0.66) CAPN1CTSBCTSLCTSSCTSK
SCHEMBL3913036 0.80 CAPN1 (0.48) CAPN1CTSBCTSLCTSSCTSK
SCHEMBL3910399 0.79 CAPN1 (0.47) CAPN1CTSBCTSLCTSSCTSK
SCHEMBL25466056 0.76 LMNA (0.54) CAPN1CTSBMMP1MMP2MMP9
SCHEMBL12943103 0.74 USP30 (0.42) CAPN1CTSBCTSLCTSSCTSK
SCHEMBL3917869 0.73 CAPN1 (0.54) CAPN1CTSBMMP1MMP2MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018023054-A1 PROTEASE TRANSITION STATE INHIBITOR PRODRUGS KANSAS STATE UNIVERSITY RESEARCH FOUNDATION (US) 2018-02-01 WO disclosed