SCHEMBL19852058

SCHEMBL19852058

CC1(O)COc2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.37
CYP1A2 P05177 1/20 0.36
ABCG2 Q9UNQ0 1/20 0.36
ITGB2 P05107 1/20 0.36
ICAM1 P05362 1/20 0.36
ITGAL P20701 1/20 0.36
ALOX15 P16050 1/20 0.36
CHRNB2 P17787 1/20 0.35
SLC6A2 P23975 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNA4 P43681 1/20 0.35
SLC6A3 Q01959 1/20 0.35
CHRM3 P20309 1/20 0.35
TAAR1 Q96RJ0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14031240 0.85 TAAR1 (0.34) AKR1B1ABCG2ITGB2ICAM1ITGAL
SCHEMBL30403463 0.80 ITGB2 (0.43) ITGB2ICAM1ITGAL
SCHEMBL321566 0.78 NOTUM (0.42) ABCG2ITGB2ICAM1ITGALTAAR1
SCHEMBL7031384 0.77 ITGB2 (0.40) ITGB2ICAM1ITGAL
SCHEMBL14436805 0.76 CHRNA7 (0.40) AKR1B1CHRM3
SCHEMBL11156161 0.76 ABCG2 (0.46) ABCG2ITGB2ICAM1ITGALALOX15
SCHEMBL18211723 0.75 ABCG2 (0.36) ABCG2ITGB2ICAM1ITGALTAAR1
SCHEMBL25899948 0.75 HTR1A (0.42) AKR1B1SLC6A2
SCHEMBL30403909 0.73 ITGB2 (0.40) AKR1B1ITGB2ICAM1ITGAL
SCHEMBL3355781 0.73 MAP3K14 (0.35) AKR1B1ABCG2ITGB2ICAM1ITGAL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11186564-B2 Dual NAV1.2/5HT2a inhibitors for treating CNS disorders SUNOVION PHARMACEUTICALS INC. (US) 2021-11-30 US disclosed
WO-2021036514-A1 PPAR γ/δ DUAL AGONIST, PREPARATION METHOD THEREOF AND USE THEREOF IN PREPARING A DRUG 广东药科大学 2021-03-04 WO disclosed
US-20190194163-A1 DUAL NAV1.2/5HT2a INHIBITORS FOR TREATING CNS DISORDERS SUNOVION PHARMACEUTICALS INC. (US) 2019-06-27 US disclosed
WO-2018026371-A1 DUAL NAV1.2/5HT2A INHIBITORS FOR TREATING CNS DISORDERS SUNOVION PHARMACEUTICALS INC. (US) 2018-02-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190194163-A1 DUAL NAV1.2/5HT2a INHIBITORS FOR TREATING CNS DISORDERS SCN2A, HTR2A, HTR2C AKR1B1 2869/4885CYP1A2 201/4885ABCG2 418/4885
US-11186564-B2 Dual NAV1.2/5HT2a inhibitors for treating CNS disorders SCN2A, HTR2A, HTR2C AKR1B1 2869/4885CYP1A2 201/4885ABCG2 418/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.