SCHEMBL19859928

SCHEMBL19859928

CC1(C)CC(C)(C)c2c1ccc1c2cc(-c2ccccc2)c2ncccc21

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TOP1 P11387 7/20 0.38
CKS1B P61024 3/20 0.35
SKP2 Q13309 3/20 0.35
GLO1 Q04760 2/20 0.35
PDE4A P27815 3/20 0.33
PIK3CD O00329 1/20 0.32
CCR1 P32246 1/20 0.32
CCR8 P51685 1/20 0.32
PIK3R2 O00459 1/20 0.32
ALDH1A1 P00352 1/20 0.31
COMT P21964 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16582575 0.85 TOP1 (0.38) TOP1CKS1BSKP2GLO1PDE4A
SCHEMBL19859927 0.82 CCR1 (0.38) CCR1CCR8ALDH1A1COMT
SCHEMBL16582578 0.77 KDM4E (0.33) ALDH1A1
SCHEMBL16582720 0.75 KDM4E (0.43) CCR1CCR8ALDH1A1COMT
SCHEMBL14461472 0.72 TOP1 (0.50) TOP1PDE4ACCR1CCR8ALDH1A1
SCHEMBL16582736 0.71 HSP90AA1 (0.42) CCR1CCR8ALDH1A1
SCHEMBL14461484 0.70 TOP1 (0.48) TOP1PDE4ACCR1CCR8ALDH1A1
SCHEMBL16582584 0.68 CCR1 (0.37) CCR1CCR8COMT
SCHEMBL25792185 0.68 RARB (0.41) TOP1
SCHEMBL24406913 0.68 TOP1 (0.46) TOP1CKS1BSKP2GLO1PDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9893299-B2 Heterocyclic compounds MERCK PATENT GMBH (DE) 2018-02-13 US disclosed