SCHEMBL19859927

SCHEMBL19859927

Cc1cc2c3c(ccc2c2cccnc12)C(C)(C)CC3(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 3/20 0.38
CCR8 P51685 3/20 0.38
L3MBTL1 Q9Y468 3/20 0.37
NPC1 O15118 2/20 0.37
HSP90AA1 P07900 1/20 0.37
PSMD14 O00487 2/20 0.35
COPS5 Q92905 2/20 0.35
HTT P42858 2/20 0.35
SLC6A2 P23975 1/20 0.35
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
CCR5 P51681 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
PRMT5 O14744 1/20 0.33
COMT P21964 1/20 0.33
HTR1A P08908 1/20 0.33
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33
DYRK1A Q13627 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16582584 0.83 CCR1 (0.37) CCR1CCR8L3MBTL1NPC1HSP90AA1
SCHEMBL19859928 0.82 TOP1 (0.38) CCR1CCR8COMTALDH1A1
SCHEMBL16582720 0.79 KDM4E (0.43) CCR1CCR8L3MBTL1NPC1HSP90AA1
SCHEMBL16582736 0.71 HSP90AA1 (0.42) CCR1CCR8L3MBTL1NPC1HSP90AA1
SCHEMBL19859933 0.69
SCHEMBL16582575 0.67 TOP1 (0.38) CCR1CCR8CCR5COMT
SCHEMBL16582618 0.67 OPRK1 (0.32) KMT2AMAPT
SCHEMBL16582562 0.66 CCR1 (0.31) CCR1CCR8CCR5
SCHEMBL19859936 0.66 CCR1 (0.36) CCR1CCR8L3MBTL1NPC1HSP90AA1
SCHEMBL17173759 0.66 KDM4E (0.52) CCR1CCR8L3MBTL1NPC1HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9893299-B2 Heterocyclic compounds MERCK PATENT GMBH (DE) 2018-02-13 US disclosed