SCHEMBL19860190

SCHEMBL19860190

C=CC(=O)Nc1cc(Nc2nc(C3=CCCCC3)c3cc[nH]c3n2)c(OC)cc1N1CCN(C)CC1

nearest known ligand 0.73

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
EGFR P00533 19/20 0.73
IGF1R P08069 2/20 0.54
KCNH2 Q12809 2/20 0.54
JAK3 P52333 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19860191 0.86 EGFR (0.82) EGFRIGF1RKCNH2JAK3
SCHEMBL19239592 0.84 EGFR (0.82) EGFRIGF1RKCNH2
SCHEMBL17467217 0.84 EGFR (1.00) EGFRIGF1RKCNH2
SCHEMBL19860187 0.84 EGFR (0.72) EGFRIGF1RKCNH2JAK3
SCHEMBL19860192 0.83 EGFR (0.80) EGFRIGF1RKCNH2
SCHEMBL19860792 0.83 EGFR (0.70) EGFRIGF1RKCNH2JAK3
SCHEMBL19860193 0.82 EGFR (0.73) EGFRIGF1RKCNH2
SCHEMBL17467214 0.81 EGFR (0.75) EGFRIGF1RKCNH2
SCHEMBL19860188 0.81 EGFR (0.76) EGFRIGF1RKCNH2
SCHEMBL17467224 0.81 EGFR (0.69) EGFRIGF1RKCNH2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9890168-B2 2,4-disubstituted 7H-pyrrolo[2,3-d]pyrimidine derivative, preparation method and medicinal use thereof SHANGHAI HAIYAN PHARMACEUTICAL TECHNOLOGY CO., LTD. (CN) 2018-02-13 US disclosed
US-9890168-B2 2,4-disubstituted 7H-pyrrolo[2,3-d]pyrimidine derivative, preparation method and medicinal use thereof SHANGHAI HAIYAN PHARMACEUTICAL TECHNOLOGY CO., LTD. (CN) 2018-02-13 US disclosed