SCHEMBL19861027

SCHEMBL19861027

CCc1c(F)cc(N2CCOCC2)cc1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.46
PIK3C2B O00750 3/20 0.46
ALDH1A1 P00352 5/20 0.42
HSD17B10 Q99714 4/20 0.42
MEN1 O00255 4/20 0.42
KMT2A Q03164 4/20 0.42
MAPT P10636 3/20 0.42
HPGD P15428 2/20 0.42
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
LMNA P02545 2/20 0.41
MYC P01106 1/20 0.41
WDR5 P61964 1/20 0.41
ALOX15 P16050 2/20 0.41
HTT P42858 2/20 0.41
USP2 O75604 1/20 0.41
TP53 P04637 1/20 0.41
MAPK1 P28482 1/20 0.41
NPC1 O15118 2/20 0.40
NUDT1 P36639 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28991001 0.82 KDM4E (0.42) KDM4EPIK3C2BALDH1A1HSD17B10MEN1
SCHEMBL16922688 0.79 KDM4E (0.55) KDM4EPIK3C2BALDH1A1HSD17B10MEN1
SCHEMBL28123984 0.79 PRKDC (0.48) KDM4EALDH1A1MAPTHPGDTDP1
SCHEMBL22657488 0.78 AKR1C3 (0.42) KDM4EALDH1A1MEN1KMT2AMAPT
SCHEMBL27410032 0.78 MYC (0.43) KDM4EPIK3C2BALDH1A1HSD17B10MEN1
SCHEMBL12831239 0.76 KDM4E (0.44) KDM4EALDH1A1HSD17B10MEN1KMT2A
SCHEMBL28991680 0.76 KDM4E (0.46) KDM4EALDH1A1HSD17B10MEN1KMT2A
SCHEMBL20467558 0.76 KDM4E (0.50) KDM4EALDH1A1HSD17B10MEN1KMT2A
SCHEMBL2376896 0.76 LGMN (0.49) KDM4EALDH1A1HSD17B10MEN1KMT2A
SCHEMBL22996752 0.75 KDM4E (0.50) KDM4EPIK3C2BALDH1A1HSD17B10MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023220741-A1 ALPHA 4 BETA 7 INTEGRIN MODULATORS AND USES THEREOF DICE MOLECULES SV, INC. (US) 2023-11-16 WO disclosed
US-9890119-B2 Indole and azaindole derivative having AMPK-activating activity SHIONOGI & CO., LTD. (JP) 2018-02-13 US disclosed