SCHEMBL19863553

SCHEMBL19863553

O=S1(=O)CC2(CCCCC2)C1

nearest known ligand 0.35

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21782681 0.97
SCHEMBL16768934 0.90
SCHEMBL16545185 0.79 LMNA (0.31)
SCHEMBL3137029 0.75
SCHEMBL21782682 0.75
SCHEMBL19971177 0.71 ALDH1A1 (0.30)
SCHEMBL1812050 0.71
SCHEMBL31017583 0.71 ALDH1A1 (0.30)
SCHEMBL8763394 0.71 ALDH1A1 (0.30)
SCHEMBL1003911 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11396512-B2 CDK2/4/6 inhibitors PFIZER INC. (US) 2022-07-26 US disclosed
US-20220089580-A1 CYCLIN DEPENDENT KINASE INHIBITORS PFIZER INC. (US) 2022-03-24 US disclosed
US-11220494-B2 Cyclin dependent kinase inhibitors PFIZER INC. (US) 2022-01-11 US disclosed
US-20200392142-A1 CDK2/4/6 Inhibitors PFIZER INC. (US) 2020-12-17 US disclosed
US-20200354350-A1 CYCLIN DEPENDENT KINASE INHIBITORS PFIZER INC. (US) 2020-11-12 US disclosed
US-10800783-B2 CDK2/4/6 inhibitors PFIZER INC. (US) 2020-10-13 US disclosed
US-10766884-B2 Cyclin dependent kinase inhibitors PFIZER INC. (US) 2020-09-08 US disclosed
EP-3617204-A1 INDOLEAMINE 2,3-DIOXYGENASE INHIBITOR AND APPLICATION Nanjing Transthera Biosciences Co. Ltd. (CN) 2020-03-04 EP disclosed
US-20190330196-A1 CYCLIN DEPENDENT KINASE INHIBITORS PFIZER INC. (US) 2019-10-31 US disclosed
US-20190135817-A1 CDK2/4/6 Inhibitors PFIZER INC. (US) 2019-05-09 US disclosed
US-10233188-B2 CDK2/4/6 inhibitors PFIZER INC. (US) 2019-03-19 US disclosed
WO-2018033815-A1 PYRIDOPYRIMDINONE CDK2/4/6 INHIBITORS PFIZER INC. (US) 2018-02-22 WO disclosed
US-20180044344-A1 CDK2/4/6 Inhibitors PFIZER INC. (US) 2018-02-15 US disclosed
US-20180044344-A1 CDK2/4/6 Inhibitors PFIZER INC. (US) 2018-02-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (11 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10766884-B2 Cyclin dependent kinase inhibitors CCNY, CCNI, CCNK TSHR 2494/4885CYP2C19 3286/4885
US-20200354350-A1 CYCLIN DEPENDENT KINASE INHIBITORS CCNY, CCNI, CCNK TSHR 2494/4885CYP2C19 3286/4885
US-20200392142-A1 CDK2/4/6 Inhibitors CDK2, CDK6, CDK20 TSHR 1117/4885CYP2C19 1039/4885
US-11396512-B2 CDK2/4/6 inhibitors CDK2, CDK6, CDK20 TSHR 1070/4885CYP2C19 1040/4885
US-10800783-B2 CDK2/4/6 inhibitors CDK2, CDK6, CDK20 TSHR 1070/4885CYP2C19 1040/4885
US-20180044344-A1 CDK2/4/6 Inhibitors CDK2, CDK6, CDK20 TSHR 1070/4885CYP2C19 1040/4885
US-20190330196-A1 CYCLIN DEPENDENT KINASE INHIBITORS CCNY, CCNI, CCNK TSHR 2494/4885CYP2C19 3286/4885
US-20190135817-A1 CDK2/4/6 Inhibitors CDK2, CDK6, CDK20 TSHR 1070/4885CYP2C19 1040/4885
US-10233188-B2 CDK2/4/6 inhibitors CDK2, CDK6, CDK20 TSHR 1070/4885CYP2C19 1040/4885
US-11220494-B2 Cyclin dependent kinase inhibitors CCNY, CCNI, CCNK TSHR 2494/4885CYP2C19 3286/4885
US-20220089580-A1 CYCLIN DEPENDENT KINASE INHIBITORS CCNY, CCNI, CCNK TSHR 2494/4885CYP2C19 3286/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.