SCHEMBL19866041

SCHEMBL19866041

CC1Cc2c([nH]c3cc(F)ccc23)C(C(=O)OC(=O)c2ccc(F)cc2)=CN1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 12/20 0.40
PARP1 P09874 1/20 0.36
MAP2K4 P45985 1/20 0.36
TUBB4A P04350 1/20 0.35
TUBB P07437 1/20 0.35
TUBA3C P0DPH7 1/20 0.35
TUBA1B P68363 1/20 0.35
TUBA4A P68366 1/20 0.35
TUBB4B P68371 1/20 0.35
TUBB3 Q13509 1/20 0.35
TUBB2A Q13885 1/20 0.35
TUBB8 Q3ZCM7 1/20 0.35
TUBA3E Q6PEY2 1/20 0.35
TUBA1A Q71U36 1/20 0.35
TUBA1C Q9BQE3 1/20 0.35
TUBB6 Q9BUF5 1/20 0.35
TUBB2B Q9BVA1 1/20 0.35
TUBB1 Q9H4B7 1/20 0.35
MAPKAPK2 P49137 1/20 0.34
MEN1 O00255 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4441689 0.91 NR1H4 (0.49) NR1H4TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL688263 0.84 KMT2A (0.38) PARP1MAP2K4TUBB4ATUBBTUBA3C
SCHEMBL273508 0.83 NR1H4 (0.49) NR1H4
SCHEMBL29881710 0.71 NR1H4 (0.44) NR1H4
SCHEMBL278969 0.70 NR1H4 (0.58) NR1H4MEN1KMT2AKCNH2
SCHEMBL273651 0.70 NR1H4 (0.51) NR1H4MEN1KMT2A
SCHEMBL29880972 0.69 NR1H4 (0.59) NR1H4
SCHEMBL273595 0.68 NR1H4 (0.52) NR1H4MEN1KMT2A
SCHEMBL273035 0.65 NR1H4 (0.53) NR1H4MEN1KMT2A
SCHEMBL19866042 0.65 TUBB4A (0.36) NR1H4PARP1MAP2K4TUBB4ATUBB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9895380-B2 Methods and pharmaceutical compositions for the treatment of hepatitis B virus infection INSERM (INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE) (FR) 2018-02-20 US disclosed