SCHEMBL19881908

SCHEMBL19881908

NCCNc1ccc2[nH]cnc2n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.39
HRH3 Q9Y5N1 1/20 0.37
KDM4E B2RXH2 1/20 0.35
HRH4 Q9H3N8 1/20 0.35
CDK2 P24941 3/20 0.35
PIM1 P11309 5/20 0.34
PIM2 Q9P1W9 4/20 0.34
TLR9 Q9NR96 1/20 0.34
TLR8 Q9NR97 1/20 0.34
TLR7 Q9NYK1 1/20 0.34
MAPK14 Q16539 1/20 0.34
CDK7 P50613 2/20 0.34
CDK9 P50750 2/20 0.34
CDC7 O00311 1/20 0.34
DAPK3 O43293 1/20 0.34
ROCK2 O75116 1/20 0.34
PRKD3 O94806 1/20 0.34
MAP4K4 O95819 1/20 0.34
PAK4 O96013 1/20 0.34
PRKACA P17612 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21295271 0.75 CYP1A2 (0.50) ALDH1A1KDM4ECDK2MAPK14MAP4K4
SCHEMBL1998243 0.70 ALDH1A1 (0.37) ALDH1A1KDM4ECDK2MAPK14CDK7
SCHEMBL1998246 0.70 ALDH1A1 (0.37) ALDH1A1KDM4ECDK2MAPK14CDK7
SCHEMBL19881862 0.70 NPSR1 (0.37) ALDH1A1KDM4EPIM1PIM2TLR9
SCHEMBL13256589 0.69 CDK2 (0.60) ALDH1A1KDM4ECDK2PIM1PIM2
SCHEMBL17776969 0.68 HTR1F (0.47)
SCHEMBL19881892 0.68 CHEK1 (0.47) ALDH1A1KDM4EPIM1PIM2PIM3
SCHEMBL17776531 0.68 GDA (0.46) KDM4EROCK2ROCK1
SCHEMBL19881886 0.68 PIM1 (0.49) PIM1PIM2TLR9TLR8TLR7
SCHEMBL3180578 0.67 ALDH1A1 (0.53) ALDH1A1KDM4ECDK2MAPK14CDK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3284743-B1 HETEROCYCLIC-IMIDAZOLE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS THEREOF, PREPARATION METHOD THEREFOR AND USE THEREOF SHANGHAI HUILUN LIFE SCIENCE & TECH CO LTD (CN) 2022-07-06 EP disclosed
EP-3284743-A1 HETEROCYCLIC-IMIDAZOLE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS THEREOF, PREPARATION METHOD THEREFOR AND USE THEREOF Shanghai Huilun Life Science & Technology Co., Ltd (CN) 2018-02-21 EP disclosed