Ammonia Solution, Strong

Ammonia Solution, Strong

SCHEMBL19894166

COc1cccc(CC2=NN([C@@H](Cc3ccc([N+](=O)[O-])cc3)c3csc(-c4cccs4)n3)CS2)c1.N

nearest known ligand 0.35

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.35
ADORA3 P0DMS8 1/20 0.35
ADORA2B P29275 1/20 0.35
ADORA1 P30542 1/20 0.35
MEN1 O00255 6/20 0.34
KMT2A Q03164 6/20 0.34
ALDH1A1 P00352 6/20 0.34
MAPT P10636 3/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
POLB P06746 1/20 0.34
CRHBP P24387 1/20 0.34
CRHR2 Q13324 1/20 0.34
HTT P42858 1/20 0.33
FPR1 P21462 1/20 0.33
FPR2 P25090 1/20 0.33
USP2 O75604 4/20 0.33
CYP1A2 P05177 4/20 0.33
CYP3A4 P08684 4/20 0.33
CASP1 P29466 4/20 0.33
CASP7 P55210 4/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL870698 0.75 PTPRB (0.57) ADORA2AADORA3ADORA2BADORA1MEN1
SCHEMBL4009024 0.75 PTPRB (0.57) ADORA2AADORA3ADORA2BADORA1MEN1
SCHEMBL686535 0.71 MAPT (0.47) MEN1KMT2AALDH1A1MAPTSMN1; SMN2
SCHEMBL16573552 0.70 MEN1 (0.43) MEN1KMT2AALDH1A1MAPTHTT
SCHEMBL28293150 0.70 ALDH1A1 (0.35) ADORA2AMEN1KMT2AALDH1A1MAPT
SCHEMBL28293151 0.70 ALDH1A1 (0.35) ADORA2AMEN1KMT2AALDH1A1MAPT
SCHEMBL23303560 0.70 PTPRB (0.46) MEN1KMT2AALDH1A1MAPTHTT
SCHEMBL8587434 0.70 PTPRB (0.46) MEN1KMT2AALDH1A1MAPTHTT
SCHEMBL23304230 0.69 MEN1 (0.43) MEN1KMT2AALDH1A1MAPTSMN1; SMN2
SCHEMBL23304233 0.69 MEN1 (0.43) MEN1KMT2AALDH1A1MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3287455-A1 HUMAN PROTEIN TYROSINE PHOSPHATASE INHIBITORS AND METHODS OF USE Aerpio Therapeutics, Inc. (US) 2018-02-28 EP disclosed