SCHEMBL19902371

SCHEMBL19902371

CCCCC[C@H](C)c1n[nH]c(=O)c2ccccc12

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.54
POLB P06746 3/20 0.54
HTT P42858 2/20 0.44
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.43
ALDH1A1 P00352 2/20 0.43
PRMT5 O14744 1/20 0.42
CYP1A2 P05177 1/20 0.42
ATM Q13315 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
AR P10275 5/20 0.40
PARP1 P09874 1/20 0.40
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9229130 0.81 KDM4E (0.39) TSHRKMT2AMEN1ALDH1A1CYP1A2
SCHEMBL17354960 0.79 TSHR (0.56) TSHRPOLBHTTKMT2AMEN1
SCHEMBL25310697 0.79 POLB (0.63) TSHRPOLBHTTKMT2AMEN1
SCHEMBL25310041 0.77 TSHR (0.67) TSHRPOLBHTTKMT2AMEN1
SCHEMBL17354964 0.77 TSHR (0.53) TSHRPOLBHTTKMT2AMEN1
SCHEMBL1786764 0.76 POLB (0.68) TSHRPOLBHTTKMT2AMEN1
SCHEMBL29480990 0.76 POLB (0.68) TSHRPOLBHTTKMT2AMEN1
SCHEMBL13265507 0.75 POLB (0.55) TSHRPOLBHTTKMT2AMEN1
SCHEMBL28857250 0.73 PRMT5 (0.58) POLBSMN1; SMN2ALDH1A1PRMT5AR
SCHEMBL19902401 0.72 POLB (0.51) TSHRPOLBHTTKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9902702-B2 Spirocycloheptanes as inhibitors of rock BRISTOL-MYERS SQUIBB COMPANY (US) 2018-02-27 US disclosed