SCHEMBL19902387

SCHEMBL19902387

CCC(=O)c1nnn(-c2ccccc2OC)c1C

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 10/20 0.52
PTGS2 P35354 1/20 0.49
TP53 P04637 1/20 0.47
ALOX12 P18054 1/20 0.47
MAPT P10636 2/20 0.47
ALDH1A1 P00352 1/20 0.46
HSD11B1 P28845 1/20 0.46
SLC5A1 P13866 1/20 0.44
SLC5A2 P31639 1/20 0.44
KCNN4 O15554 1/20 0.44
HTT P42858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15897945 0.86 TP53 (0.66) NR1I2TP53ALOX12MAPTALDH1A1
SCHEMBL17454344 0.85 MAPT (0.61) NR1I2PTGS2MAPTALDH1A1KCNN4
SCHEMBL3406092 0.85 HTT (0.61) NR1I2TP53ALOX12MAPTALDH1A1
SCHEMBL17452650 0.82 NR1I2 (0.50) NR1I2MAPTALDH1A1SLC5A1SLC5A2
SCHEMBL19997265 0.81 PTGS2 (0.51) PTGS2TP53ALOX12MAPTALDH1A1
SCHEMBL20229575 0.79 NR1I2 (0.54) NR1I2ALDH1A1
SCHEMBL7988852 0.74 NR1I2 (0.56) NR1I2
SCHEMBL18172023 0.74 MAPT (0.57) NR1I2TP53MAPTALDH1A1HSD11B1
SCHEMBL20162992 0.74 NPC1 (0.52) PTGS2TP53MAPTALDH1A1
SCHEMBL30038295 0.74 NPC1 (0.52) PTGS2TP53MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9902702-B2 Spirocycloheptanes as inhibitors of rock BRISTOL-MYERS SQUIBB COMPANY (US) 2018-02-27 US disclosed