SCHEMBL19902544

SCHEMBL19902544

CCC(=O)c1sc(N2CCOCC2)nc1C

nearest known ligand 0.72

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 4/20 0.72
PIK3CB P42338 4/20 0.72
PIK3CA P42336 2/20 0.72
ALDH1A1 P00352 6/20 0.69
GAA P10253 3/20 0.69
KDM4E B2RXH2 1/20 0.69
MAPT P10636 1/20 0.69
SMN1; SMN2 Q16637 1/20 0.69
ALOX5 P09917 3/20 0.44
PTGS2 P35354 2/20 0.43
HPGD P15428 1/20 0.42
AR P10275 2/20 0.41
PIK3CG P48736 3/20 0.41
HTT P42858 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CNR1 P21554 1/20 0.40
NUDT1 P36639 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6120595 0.87 PIK3CD (0.70) PIK3CDPIK3CBPIK3CAALDH1A1GAA
SCHEMBL20229568 0.87 PIK3CD (0.52) PIK3CDPIK3CBPIK3CAALDH1A1GAA
Bromide SCHEMBL6114011 0.86 PIK3CD (0.68) PIK3CDPIK3CBPIK3CAALDH1A1GAA
SCHEMBL1574758 0.84 PIK3CD (0.78) PIK3CDPIK3CBPIK3CAALDH1A1GAA
SCHEMBL3328268 0.84 PIK3CD (1.00) PIK3CDPIK3CBPIK3CAALDH1A1GAA
SCHEMBL625865 0.83 PIK3CA (0.68) PIK3CDPIK3CBPIK3CAALDH1A1GAA
SCHEMBL3328174 0.82 PIK3CD (0.76) PIK3CDPIK3CBPIK3CAALDH1A1GAA
Hydrochloric Acid SCHEMBL6114749 0.82 PIK3CD (0.76) PIK3CDPIK3CBPIK3CAALDH1A1GAA
SCHEMBL24829791 0.82 ALDH1A1 (1.00) PIK3CDPIK3CBPIK3CAALDH1A1GAA
Hydrochloric Acid SCHEMBL5010640 0.81 PIK3CD (0.74) PIK3CDPIK3CBPIK3CAALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9902702-B2 Spirocycloheptanes as inhibitors of rock BRISTOL-MYERS SQUIBB COMPANY (US) 2018-02-27 US disclosed