SCHEMBL19902597

SCHEMBL19902597

CCC(=O)c1cnn2cc(COC)ccc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.38
RAB9A P51151 4/20 0.38
SMN1; SMN2 Q16637 4/20 0.38
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
KLF5 Q13887 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
KDM4E B2RXH2 4/20 0.34
ALDH1A1 P00352 4/20 0.34
EPHB3 P54753 2/20 0.34
HSD17B10 Q99714 1/20 0.34
PDE2A O00408 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
FFAR4 Q5NUL3 1/20 0.33
HTT P42858 2/20 0.33
HSP90AB1 P08238 1/20 0.33
IRAK4 Q9NWZ3 2/20 0.32
MAPT P10636 1/20 0.32
HAT1 O14929 2/20 0.32
EP300 Q09472 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17454509 0.87 NPC1 (0.40) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL25369434 0.86 PTPN1 (0.37) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL25365640 0.85 SMN1; SMN2 (0.41) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL17452740 0.83 HAT1 (0.37) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL19997307 0.81 MEN1 (0.43) RAB9ASMN1; SMN2KMT2AMEN1KDM4E
SCHEMBL19902430 0.78 NPC1 (0.36) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL19902685 0.78 NPC1 (0.38) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL19902395 0.77 THRA (0.37) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL31547045 0.76 NPC1 (0.48) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL19902366 0.76 MAPT (0.46) RAB9ASMN1; SMN2KMT2AMEN1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9902702-B2 Spirocycloheptanes as inhibitors of rock BRISTOL-MYERS SQUIBB COMPANY (US) 2018-02-27 US disclosed