SCHEMBL19902430

SCHEMBL19902430

CCC(=O)c1cnn2cc(CCC(F)(F)F)ccc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
KLF5 Q13887 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
KDM4E B2RXH2 3/20 0.33
ALDH1A1 P00352 3/20 0.33
HTT P42858 2/20 0.33
ROCK2 O75116 1/20 0.33
EPHB3 P54753 3/20 0.33
PDE2A O00408 1/20 0.33
HAT1 O14929 6/20 0.33
EP300 Q09472 6/20 0.33
L3MBTL1 Q9Y468 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32
KCNH2 Q12809 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17454523 0.88 NPC1 (0.38) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL19127961 0.86 SMN1; SMN2 (0.36) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL17452737 0.84 HAT1 (0.37) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL19902685 0.80 NPC1 (0.38) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL20654123 0.80 ROCK2 (0.49) RAB9AROCK2PDE2A
SCHEMBL19902395 0.79 THRA (0.37) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL20646991 0.79 ROCK2 (0.45) ROCK2PDE2APTGDR2KCNH2
SCHEMBL19902597 0.78 NPC1 (0.38) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL19902424 0.73 CCNC (0.35) MEN1KMT2AALDH1A1HTR2AHTR2C
SCHEMBL19997307 0.72 MEN1 (0.43) RAB9ASMN1; SMN2MEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9902702-B2 Spirocycloheptanes as inhibitors of rock BRISTOL-MYERS SQUIBB COMPANY (US) 2018-02-27 US disclosed