SCHEMBL19902669

SCHEMBL19902669

CCCC(=O)c1nn(C)c2ccccc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.56
TSHR P16473 2/20 0.55
HTR3E A5X5Y0 2/20 0.49
HTR3B O95264 2/20 0.49
HTR3A P46098 2/20 0.49
HTR3D Q70Z44 2/20 0.49
HTR3C Q8WXA8 2/20 0.49
ELANE P08246 3/20 0.48
F2 P00734 1/20 0.48
PLAU P00749 1/20 0.48
ALDH1A1 P00352 1/20 0.47
CYP3A4 P08684 1/20 0.47
MAPK1 P28482 1/20 0.47
HSD17B10 Q99714 1/20 0.47
HDAC3 O15379 1/20 0.46
HDAC1 Q13547 1/20 0.46
SLC22A2 O15244 1/20 0.45
CHRNB2 P17787 1/20 0.45
CHRNA3 P32297 1/20 0.45
CHRNA4 P43681 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19902668 0.89 KDM4E (0.57) KDM4ETSHRHTR3EHTR3BHTR3A
SCHEMBL18313403 0.85 KDM4E (0.57) KDM4ETSHRHTR3EHTR3BHTR3A
Maleic Acid SCHEMBL9775796 0.81 KDM4E (0.54) KDM4ETSHRHTR3EHTR3BHTR3A
Fumaric Acid SCHEMBL9775801 0.81 KDM4E (0.54) KDM4ETSHRHTR3EHTR3BHTR3A
Fumaric Acid SCHEMBL9775792 0.81 KDM4E (0.54) KDM4ETSHRHTR3EHTR3BHTR3A
SCHEMBL6858031 0.80 KDM4E (0.56) KDM4ETSHRHTR3EHTR3BHTR3A
SCHEMBL496589 0.80 KDM4E (0.62) KDM4ETSHRHTR3EHTR3BHTR3A
SCHEMBL30467838 0.80 KDM4E (0.62) KDM4ETSHRHTR3EHTR3BHTR3A
SCHEMBL30251861 0.80 KDM4E (0.62) KDM4ETSHRHTR3EHTR3BHTR3A
SCHEMBL7297926 0.80 KDM4E (0.62) KDM4ETSHRHTR3EHTR3BHTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9902702-B2 Spirocycloheptanes as inhibitors of rock BRISTOL-MYERS SQUIBB COMPANY (US) 2018-02-27 US disclosed