SCHEMBL19902723

SCHEMBL19902723

CC[C@]1(CCc2n[nH]c(=O)c3ccccc23)C[C@H](NC(=O)c2ccc(-c3cn[nH]c3)cc2OC)C1

nearest known ligand 0.46

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 19/20 0.46
ROCK1 Q13464 19/20 0.46
PARP1 P09874 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19902379 0.87 ROCK2 (0.52) ROCK2ROCK1
SCHEMBL20229914 0.86 ROCK2 (0.44) ROCK2ROCK1PARP1
SCHEMBL19902407 0.81 ROCK2 (0.51) ROCK2ROCK1
SCHEMBL17452930 0.81 ROCK2 (0.56) ROCK2ROCK1
SCHEMBL19902635 0.79 ROCK2 (0.45) ROCK2ROCK1
SCHEMBL19902719 0.78 ROCK2 (0.52) ROCK2ROCK1
SCHEMBL20229925 0.74 PARP1 (0.41) ROCK2ROCK1PARP1
SCHEMBL20229895 0.74 PARP1 (0.41) ROCK2PARP1
SCHEMBL20229939 0.73 BRD4 (0.39) ROCK2PARP1
SCHEMBL19902509 0.72 USP30 (0.46) ROCK2ROCK1PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9902702-B2 Spirocycloheptanes as inhibitors of rock BRISTOL-MYERS SQUIBB COMPANY (US) 2018-02-27 US disclosed