SCHEMBL19902407

SCHEMBL19902407

CC[C@]1(CCc2n[nH]c(=O)c3ccccc23)C[C@H](NC(=O)c2ccc(-c3cn[nH]c3)c(C)c2)C1

nearest known ligand 0.51

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 20/20 0.51
ROCK1 Q13464 20/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19902379 0.92 ROCK2 (0.52) ROCK2ROCK1
SCHEMBL19902635 0.90 ROCK2 (0.45) ROCK2ROCK1
SCHEMBL20229914 0.89 ROCK2 (0.44) ROCK2ROCK1
SCHEMBL19902723 0.81 ROCK2 (0.46) ROCK2ROCK1
SCHEMBL20229925 0.81 PARP1 (0.41) ROCK2ROCK1
SCHEMBL17452927 0.81 ROCK2 (0.55) ROCK2ROCK1
SCHEMBL20229895 0.80 PARP1 (0.41) ROCK2
SCHEMBL19902406 0.78 ROCK2 (0.61) ROCK2ROCK1
SCHEMBL20229910 0.78 CHRNA7 (0.43)
SCHEMBL19902374 0.78 ROCK2 (0.51) ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9902702-B2 Spirocycloheptanes as inhibitors of rock BRISTOL-MYERS SQUIBB COMPANY (US) 2018-02-27 US disclosed