SCHEMBL19904154

SCHEMBL19904154

C=C/C=C\c1cc(C)cnc1C

nearest known ligand 0.32

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.32
CCR5 P51681 1/20 0.32
CCR8 P51685 1/20 0.32
NOS3 P29474 1/20 0.32
NOS1 P29475 1/20 0.32
NOS2 P35228 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25129348 0.81 NOS3 (0.47) CCR1CCR5CCR8NOS3NOS1
SCHEMBL11881227 0.79 CCR1 (0.37) CCR1CCR5CCR8NOS3NOS1
SCHEMBL18634102 0.78 NOS2 (0.35) CCR1CCR5CCR8NOS3NOS1
SCHEMBL22279036 0.76 BRD4 (0.33)
SCHEMBL24466707 0.73 NOS3 (0.41) CCR1CCR5CCR8NOS3NOS1
SCHEMBL23655447 0.73 CCR1 (0.32) CCR1CCR5CCR8NOS3NOS1
SCHEMBL18391431 0.73 CYP1A2 (0.32)
SCHEMBL6626617 0.71 ERN1 (0.46) CCR1CCR5CCR8NOS3NOS1
SCHEMBL29952796 0.71 ERN1 (0.46) CCR1CCR5CCR8NOS3NOS1
SCHEMBL19415151 0.71 CCR1 (0.33) CCR1CCR5CCR8NOS3NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3287459-A1 PURINYL-N-HYDROXYL PYRIMIDINE FORMAMIDE DERIVATIVES, PREPARATION METHOD THEREFOR AND USE THEREOF Guizhou Bailing Enterprise Group Pharmaceutical Co., Ltd. (CN) 2018-02-28 EP disclosed