SCHEMBL19904593

SCHEMBL19904593

O=C(NC(Cc1cc(F)c2c(c1)OCCO2)CN1CCC1)[C@@H]1CCN(c2ccc3ccccc3c2)C1

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.36
HTR1A P08908 1/20 0.36
CAPN1 P07384 4/20 0.34
TPSAB1 Q15661 1/20 0.34
CHRM2 P08172 2/20 0.34
HDAC4 P56524 1/20 0.34
CHRM4 P08173 3/20 0.33
CCR4 P51679 1/20 0.33
BDKRB1 P46663 4/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19904561 0.98 MCHR1 (0.36) MCHR1HTR1ACAPN1TPSAB1CHRM2
SCHEMBL19904535 0.94 KDM4E (0.37) HTR1A
SCHEMBL19904324 0.94 KDM4E (0.37) HTR1A
SCHEMBL19904455 0.93 KMT2A (0.36) MCHR1HTR1ACHRM2
SCHEMBL19904590 0.93 KMT2A (0.36) MCHR1HTR1ACHRM2
SCHEMBL19904498 0.93 KDM4E (0.37) HTR1A
SCHEMBL19904488 0.89 KMT2A (0.38) HTR1ACHRM2HDAC4
SCHEMBL19904389 0.88 UGCG (0.40) HTR1ACHRM4
SCHEMBL19904542 0.88 UGCG (0.40) HTR1ACHRM4
SCHEMBL19904570 0.88 NAMPT (0.33) HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3063141-B1 N-(1-HYDROXY-3-(PYRROLIDINYL)PROPAN-2-YL)PYRROLIDINE-3-CARBOXAMIDE DERIVATIVES AS GLUCOSYLCERAMIDE SYNTHASE INHIBITORS BIOMARIN PHARM INC (US) 2018-02-28 EP disclosed