SCHEMBL19904590

SCHEMBL19904590

O=C(NC(Cc1cc(F)c2c(c1)OCCO2)CN1CCC1)C1CCN(c2ccc3cc(Cl)ccc3c2)C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.36
PROKR2 Q8NFJ6 1/20 0.36
NOTUM Q6P988 2/20 0.35
HTR1A P08908 1/20 0.35
MAPT P10636 3/20 0.34
KDM4E B2RXH2 2/20 0.34
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TP53 P04637 1/20 0.33
MAPK1 P28482 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
SSTR3 P32745 2/20 0.33
PDCD1 Q15116 1/20 0.33
CD274 Q9NZQ7 1/20 0.33
EPHX2 P34913 1/20 0.33
SSTR1 P30872 1/20 0.33
CHRM2 P08172 1/20 0.33
TRPV1 Q8NER1 1/20 0.33
MCHR1 Q99705 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19904455 1.00 KMT2A (0.36) KMT2APROKR2NOTUMHTR1AMAPT
SCHEMBL19904488 0.93 KMT2A (0.38) KMT2APROKR2NOTUMHTR1AMAPT
SCHEMBL19904324 0.93 KDM4E (0.37) NOTUMHTR1AKDM4ESSTR3SSTR1
SCHEMBL19904593 0.93 MCHR1 (0.36) HTR1ACHRM2MCHR1
SCHEMBL19904535 0.93 KDM4E (0.37) NOTUMHTR1AKDM4ESSTR3SSTR1
SCHEMBL19904427 0.92 KMT2A (0.38) KMT2APROKR2NOTUMHTR1AMAPT
SCHEMBL19904498 0.91 KDM4E (0.37) NOTUMHTR1AKDM4EALDH1A1MAPK1
SCHEMBL19904561 0.91 MCHR1 (0.36) HTR1ACHRM2MCHR1
SCHEMBL19904368 0.91 HTR1A (0.38) KMT2APROKR2NOTUMHTR1AMAPT
SCHEMBL19904551 0.91 HTR1A (0.38) KMT2APROKR2NOTUMHTR1AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3063141-B1 N-(1-HYDROXY-3-(PYRROLIDINYL)PROPAN-2-YL)PYRROLIDINE-3-CARBOXAMIDE DERIVATIVES AS GLUCOSYLCERAMIDE SYNTHASE INHIBITORS BIOMARIN PHARM INC (US) 2018-02-28 EP disclosed