SCHEMBL19904679

SCHEMBL19904679

O=C(NC(Cc1ccc2c(c1)OCCO2)CN1CCCC1)[C@@H]1CCN(c2ccc3nccnc3c2)C1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.40
NPC1 O15118 1/20 0.40
TP53 P04637 1/20 0.40
RAB9A P51151 1/20 0.40
SSTR3 P32745 5/20 0.39
L3MBTL1 Q9Y468 3/20 0.39
ALDH1A1 P00352 2/20 0.39
USP2 O75604 1/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39
HSD17B10 Q99714 1/20 0.39
KDM4E B2RXH2 3/20 0.39
ACACB O00763 5/20 0.38
SSTR1 P30872 1/20 0.38
ALK Q9UM73 1/20 0.37
KMT2A Q03164 2/20 0.37
KCNH2 Q12809 1/20 0.37
PDCD1 Q15116 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19904362 1.00 SMN1; SMN2 (0.40) SMN1; SMN2NPC1TP53RAB9ASSTR3
SCHEMBL19904589 0.92 RAB9A (0.42) SMN1; SMN2NPC1TP53RAB9ASSTR3
SCHEMBL19904412 0.92 RAB9A (0.42) SMN1; SMN2NPC1TP53RAB9ASSTR3
SCHEMBL19904584 0.91 SMN1; SMN2 (0.41) SMN1; SMN2NPC1TP53RAB9ASSTR3
SCHEMBL19904605 0.86 ALDH1A1 (0.40) SMN1; SMN2NPC1TP53RAB9ASSTR3
SCHEMBL19904464 0.86 NOTUM (0.45) SMN1; SMN2SSTR3L3MBTL1ALDH1A1USP2
SCHEMBL19904452 0.86 ALDH1A1 (0.40) SMN1; SMN2NPC1TP53RAB9ASSTR3
SCHEMBL19904425 0.86 NOTUM (0.45) SMN1; SMN2SSTR3L3MBTL1ALDH1A1USP2
SCHEMBL19904652 0.86 KMT2A (0.49) SMN1; SMN2TP53SSTR3L3MBTL1ALDH1A1
SCHEMBL18101714 0.86 KMT2A (0.49) SMN1; SMN2TP53SSTR3L3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3063141-B1 N-(1-HYDROXY-3-(PYRROLIDINYL)PROPAN-2-YL)PYRROLIDINE-3-CARBOXAMIDE DERIVATIVES AS GLUCOSYLCERAMIDE SYNTHASE INHIBITORS BIOMARIN PHARM INC (US) 2018-02-28 EP disclosed