SCHEMBL19905058

SCHEMBL19905058

CNC(=O)c1ccnc2c(CCNc3cc(-c4ccc(NC5CC5)nc4)ncn3)cccc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 7/20 0.38
CYP3A4 P08684 7/20 0.38
CYP2D6 P10635 6/20 0.38
CYP2C19 P33261 6/20 0.38
USP2 O75604 5/20 0.38
CLK4 Q9HAZ1 5/20 0.38
ALDH1A1 P00352 4/20 0.38
ALOX15 P16050 3/20 0.38
HSD17B10 Q99714 3/20 0.38
HSP90AA1 P07900 1/20 0.37
CYP2C9 P11712 3/20 0.37
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
NTRK1 P04629 1/20 0.37
SYK P43405 6/20 0.36
SLC40A1 Q9NP59 2/20 0.35
MAPK1 P28482 3/20 0.34
MAPT P10636 2/20 0.34
KDM4E B2RXH2 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19905265 0.94 SYK (0.39) CYP1A2CYP3A4CYP2D6CYP2C19USP2
SCHEMBL20373325 0.92 CYP1A2 (0.38) CYP1A2CYP3A4CYP2D6CYP2C19USP2
SCHEMBL19355574 0.91 GPR39 (0.39) CYP1A2CYP3A4CYP2D6CYP2C19USP2
SCHEMBL19819884 0.89 CYP1A2 (0.38) CYP1A2CYP3A4CYP2D6CYP2C19USP2
SCHEMBL19355542 0.89 CYP1A2 (0.39) CYP1A2CYP3A4CYP2D6CYP2C19USP2
SCHEMBL19905414 0.89 CYP1A2 (0.41) CYP1A2CYP3A4CYP2D6CYP2C19USP2
SCHEMBL19355538 0.88 CYP1A2 (0.37) CYP1A2CYP3A4CYP2D6CYP2C19USP2
SCHEMBL19355532 0.88 CYP1A2 (0.37) CYP1A2CYP3A4CYP2D6CYP2C19USP2
SCHEMBL19905370 0.88 CYP1A2 (0.38) CYP1A2CYP3A4CYP2D6CYP2C19USP2
SCHEMBL19355399 0.88 CYP1A2 (0.42) CYP1A2CYP3A4CYP2D6CYP2C19USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057959-B1 DNA-PK INHIBITORS VERTEX PHARMA (US) 2018-02-28 EP disclosed