SCHEMBL19905265

SCHEMBL19905265

CNC(=O)c1ccnc2c(CCNc3cc(-c4ccc(NC5CCN(C)CC5)nc4)ncn3)cccc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 15/20 0.39
ROCK2 O75116 1/20 0.36
ROCK1 Q13464 1/20 0.36
DYRK1A Q13627 2/20 0.36
GSK3B P49841 2/20 0.36
CLK2 P49760 1/20 0.36
CLK3 P49761 1/20 0.36
USP2 O75604 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
ALOX15 P16050 1/20 0.35
CYP2C19 P33261 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CLK4 Q9HAZ1 1/20 0.35
CHEK1 O14757 1/20 0.35
IKBKB O14920 1/20 0.35
AURKA O14965 1/20 0.35
PAK4 O96013 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19905058 0.94 CYP1A2 (0.38) SYKUSP2ALDH1A1CYP1A2CYP3A4
SCHEMBL20373325 0.89 CYP1A2 (0.38) USP2ALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL19905368 0.88 WNT1 (0.36) DYRK1AGSK3BCLK2CLK3USP2
SCHEMBL19355285 0.88 PRKDC (0.40) SYKROCK2ROCK1DYRK1AGSK3B
SCHEMBL19905140 0.87 CYP1A2 (0.37) ROCK2ROCK1DYRK1AGSK3BCLK2
SCHEMBL19355574 0.86 GPR39 (0.39) SYKROCK2ROCK1USP2ALDH1A1
SCHEMBL17634663 0.85 PRKDC (0.47) SYKROCK2ROCK1DYRK1AGSK3B
SCHEMBL19819884 0.85 CYP1A2 (0.38) USP2ALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL19355474 0.85 DYRK1A (0.39) DYRK1AGSK3BCLK2CLK3USP2
SCHEMBL19355542 0.85 CYP1A2 (0.39) ROCK2GSK3BUSP2ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057959-B1 DNA-PK INHIBITORS VERTEX PHARMA (US) 2018-02-28 EP disclosed