SCHEMBL19905147

SCHEMBL19905147

CC(c1ccnc2c1OCCO2)[C@H](C)CNc1cc(-c2cc(F)c3ncccc3c2)ncn1

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
FAAH O00519 15/20 0.35
PRKDC P78527 2/20 0.35
MAPK14 Q16539 2/20 0.31
MAPK13 O15264 1/20 0.31
MAPK12 P53778 1/20 0.31
MAPK11 Q15759 1/20 0.31
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16664964 0.92 PRKDC (0.41) FAAHPRKDCMAPK14MAPK13MAPK12
SCHEMBL17634608 0.92 PRKDC (0.41) FAAHPRKDCMAPK14MAPK13MAPK12
SCHEMBL20842620 0.91 FAAH (0.34) FAAHPRKDCMAPK14MAPK13MAPK12
SCHEMBL22838685 0.86 PRKDC (0.32) FAAHPRKDCMAPK1
SCHEMBL19905243 0.84 TRPV1 (0.39) FAAHPRKDCMAPK1
SCHEMBL17634635 0.83 PRKDC (0.40) FAAHPRKDCMAPK14MAPK1
SCHEMBL17634609 0.83 PRKDC (0.43) FAAHPRKDCMAPK1
SCHEMBL19905345 0.83 FAAH (0.38) FAAHPRKDC
SCHEMBL18627044 0.82 PRKDC (0.40) FAAHPRKDCMAPK1
SCHEMBL17874642 0.82 PRKDC (0.40) FAAHPRKDC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057959-B1 DNA-PK INHIBITORS VERTEX PHARMA (US) 2018-02-28 EP disclosed