SCHEMBL19905243

SCHEMBL19905243

CC(c1ccnc2c1OCCO2)[C@H](C)CNc1cc(-c2ccc3cccnc3c2)ncn1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 2/20 0.39
FAAH O00519 13/20 0.35
PRMT5 O14744 2/20 0.35
WDR77 Q9BQA1 2/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TP53 P04637 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
HPGD P15428 1/20 0.35
ALOX15 P16050 1/20 0.35
MAPK1 P28482 1/20 0.35
CYP2C19 P33261 1/20 0.35
CLK1 P49759 1/20 0.35
DYRK1A Q13627 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CLK4 Q9HAZ1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17634599 0.91 TRPV1 (0.40) TRPV1FAAHPRMT5WDR77KDM4E
SCHEMBL22838651 0.86 TRPV1 (0.41) TRPV1FAAHPRMT5WDR77KDM4E
SCHEMBL15343256 0.84 PRKDC (0.39) TRPV1FAAHKDM4EALDH1A1TP53
SCHEMBL19905147 0.84 FAAH (0.35) FAAHMAPK1PRKDC
SCHEMBL17634610 0.81 PRKDC (0.39) FAAHKDM4EALDH1A1TP53CYP1A2
SCHEMBL19355124 0.81 PRKDC (0.39) FAAHKDM4EALDH1A1TP53CYP1A2
SCHEMBL19355264 0.80 TRPV1 (0.42) TRPV1PRMT5WDR77KDM4EALDH1A1
SCHEMBL22838638 0.80 PRKDC (0.35) FAAHKDM4EALDH1A1TP53CYP1A2
SCHEMBL22838448 0.79 TLR9 (0.36) FAAHKDM4EALDH1A1TP53CYP1A2
SCHEMBL20373242 0.79 PRKDC (0.37) TRPV1FAAHKDM4EALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057959-B1 DNA-PK INHIBITORS VERTEX PHARMA (US) 2018-02-28 EP disclosed