SCHEMBL19905368

SCHEMBL19905368

CNC(=O)c1ccnc2c(CCNc3cc(-c4ccc(N(C)C5CCN(C)CC5)nc4)ncn3)cccc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
WNT1 P04628 3/20 0.36
GSK3B P49841 3/20 0.36
DYRK1A Q13627 3/20 0.36
PIK3CD O00329 2/20 0.36
CLK4 Q9HAZ1 7/20 0.35
CYP1A2 P05177 6/20 0.35
CYP3A4 P08684 5/20 0.35
USP2 O75604 4/20 0.35
CYP2C19 P33261 3/20 0.35
CLK2 P49760 1/20 0.35
CLK3 P49761 1/20 0.35
ALDH1A1 P00352 7/20 0.34
ALOX15 P16050 4/20 0.34
CYP2D6 P10635 4/20 0.34
HSD17B10 Q99714 3/20 0.34
TBK1 Q9UHD2 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
MAPK7 Q13164 1/20 0.33
CYP2C9 P11712 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19905265 0.88 SYK (0.39) GSK3BDYRK1ACLK4CYP1A2CYP3A4
SCHEMBL19905408 0.86 CLK4 (0.37) DYRK1ACLK4CYP1A2CYP3A4USP2
SCHEMBL17634662 0.86 PRKDC (0.47) WNT1GSK3BDYRK1APIK3CDCLK4
SCHEMBL19905140 0.85 CYP1A2 (0.37) WNT1GSK3BDYRK1ACLK4CYP1A2
SCHEMBL19355474 0.85 DYRK1A (0.39) WNT1GSK3BDYRK1ACLK4CYP1A2
SCHEMBL19819884 0.84 CYP1A2 (0.38) CLK4CYP1A2CYP3A4USP2CYP2C19
SCHEMBL19905058 0.83 CYP1A2 (0.38) CLK4CYP1A2CYP3A4USP2CYP2C19
SCHEMBL19355439 0.82 USP2 (0.37) CLK4CYP1A2CYP3A4USP2CYP2C19
SCHEMBL19355532 0.82 CYP1A2 (0.37) CLK4CYP1A2CYP3A4USP2CYP2C19
SCHEMBL19905196 0.82 CLK4 (0.39) GSK3BCLK4CYP1A2CYP3A4USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057959-B1 DNA-PK INHIBITORS VERTEX PHARMA (US) 2018-02-28 EP disclosed