SCHEMBL19905490

SCHEMBL19905490

CNC(=O)c1c(F)cnc2c(C(C)CNc3cc(-c4cnc(N(C)C5CCN(CC(F)(F)F)CC5)nc4)ncn3)cccc12

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PRKDC P78527 2/20 0.41
HPGDS O60760 4/20 0.36
FAAH O00519 7/20 0.34
SOS1 Q07889 1/20 0.33
ITGB2 P05107 2/20 0.32
ICAM1 P05362 2/20 0.32
ITGAL P20701 2/20 0.32
CDK1 P06493 1/20 0.32
CDK4 P11802 1/20 0.32
CDK6 Q00534 1/20 0.32
SCN1A P35498 1/20 0.32
SCN8A Q9UQD0 1/20 0.32
TRPV4 Q9HBA0 1/20 0.32
BDKRB1 P46663 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17874743 1.00 PRKDC (0.41) PRKDCHPGDSFAAHSOS1ITGB2
SCHEMBL19905500 0.94 HPGDS (0.35) PRKDCHPGDSFAAHSOS1ITGB2
SCHEMBL17874752 0.94 PRKDC (0.40) PRKDCHPGDSFAAHSOS1ITGB2
SCHEMBL17874793 0.93 PRKDC (0.42) PRKDCFAAHITGB2ICAM1ITGAL
SCHEMBL17874725 0.92 PRKDC (0.42) PRKDCFAAHSOS1SCN1ASCN8A
SCHEMBL17874786 0.92 PRKDC (0.41) PRKDCFAAHSCN1ASCN8A
SCHEMBL17874721 0.92 PRKDC (0.43) PRKDCFAAHITGB2ICAM1ITGAL
SCHEMBL17874705 0.91 PRKDC (0.41) PRKDCHPGDSFAAHSOS1CDK1
SCHEMBL17874724 0.91 PRKDC (0.42) PRKDCFAAHSOS1ITGB2ICAM1
SCHEMBL17874723 0.89 PRKDC (0.46) PRKDCHPGDSFAAHSOS1ITGB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057959-B1 DNA-PK INHIBITORS VERTEX PHARMA (US) 2018-02-28 EP disclosed