SCHEMBL19905500

SCHEMBL19905500

CNC(=O)c1c(F)cnc2c(C(C)[C@H](C)CNc3cc(-c4cnc(N(C)C5CCN(CC(F)(F)F)CC5)nc4)ncn3)cccc12

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 4/20 0.35
PRKDC P78527 2/20 0.35
FAAH O00519 6/20 0.33
SOS1 Q07889 1/20 0.32
ITGB2 P05107 2/20 0.31
ICAM1 P05362 2/20 0.31
ITGAL P20701 2/20 0.31
CDK1 P06493 1/20 0.31
CDK4 P11802 1/20 0.31
CDK6 Q00534 1/20 0.31
EZH2 Q15910 1/20 0.31
TRPV4 Q9HBA0 1/20 0.31
BDKRB1 P46663 1/20 0.31
TBK1 Q9UHD2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19905490 0.94 PRKDC (0.41) HPGDSPRKDCFAAHSOS1ITGB2
SCHEMBL17874743 0.94 PRKDC (0.41) HPGDSPRKDCFAAHSOS1ITGB2
SCHEMBL19905336 0.91 PRKDC (0.36) PRKDCFAAHSOS1ITGB2ICAM1
SCHEMBL19905298 0.90 PRKDC (0.39) HPGDSPRKDCFAAHSOS1ITGB2
SCHEMBL19905167 0.90 HPGDS (0.35) HPGDSPRKDCFAAHSOS1CDK1
SCHEMBL17874752 0.88 PRKDC (0.40) HPGDSPRKDCFAAHSOS1ITGB2
SCHEMBL19905277 0.87 CDK1 (0.35) HPGDSPRKDCFAAHSOS1CDK1
SCHEMBL17874793 0.87 PRKDC (0.42) PRKDCFAAHITGB2ICAM1ITGAL
SCHEMBL17874725 0.86 PRKDC (0.42) PRKDCFAAHSOS1EZH2BDKRB1
SCHEMBL17874786 0.86 PRKDC (0.41) PRKDCFAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057959-B1 DNA-PK INHIBITORS VERTEX PHARMA (US) 2018-02-28 EP disclosed