SCHEMBL19905889

SCHEMBL19905889

Cc1ccnc(-c2cccc(/C(=N/N)NN)c2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.47
CNR1 P21554 1/20 0.45
CCR1 P32246 1/20 0.43
CCR5 P51681 1/20 0.43
CCR8 P51685 1/20 0.43
KARS1 Q15046 3/20 0.40
ABL1 P00519 4/20 0.39
BCR P11274 4/20 0.39
KMO O15229 2/20 0.38
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38
KMT2A Q03164 1/20 0.38
EGFR P00533 1/20 0.37
JAK2 O60674 1/20 0.36
KDR P35968 1/20 0.36
MAPK13 O15264 1/20 0.36
MAPK12 P53778 1/20 0.36
MAPK11 Q15759 1/20 0.36
MAPK14 Q16539 1/20 0.36
PLAU P00749 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20114490 0.80 PARP1 (0.48) MEN1KMT2A
SCHEMBL12408987 0.75 CYP2A6 (0.65) CYP2A6CNR1CCR1CCR5CCR8
SCHEMBL842300 0.75 PARP1 (0.61) CYP2A6CNR1CCR1CCR5CCR8
SCHEMBL23259447 0.73 CYP2A6 (0.58) CYP2A6CNR1CCR1CCR5CCR8
SCHEMBL30469353 0.72 KARS1 (0.61) CYP2A6CNR1CCR1CCR5CCR8
SCHEMBL3490679 0.72 KARS1 (0.61) CYP2A6CNR1CCR1CCR5CCR8
SCHEMBL23525600 0.72 CYP2A6 (0.57) CYP2A6CNR1CCR1CCR5CCR8
SCHEMBL30705187 0.72 CYP2A6 (0.57) CYP2A6CNR1CCR1CCR5CCR8
SCHEMBL24689981 0.72 DHODH (0.42) MEN1MAPTKMT2A
SCHEMBL2479816 0.71 CYP2A6 (0.59) CYP2A6CNR1CCR1CCR5CCR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed