SCHEMBL19905966

SCHEMBL19905966

Cc1cc2nc(-c3ccc4nc(C)n(C5CCN(C)C5)c4c3)sc2c(-c2ccc(Cl)cc2)c1CC(=O)O

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 5/20 0.36
JAK3 P52333 4/20 0.36
JAK2 O60674 2/20 0.36
IDO1 P14902 1/20 0.35
KCNH2 Q12809 1/20 0.35
MCHR1 Q99705 2/20 0.35
KDM4E B2RXH2 2/20 0.35
PTGDR2 Q9Y5Y4 2/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
KMT2A Q03164 1/20 0.34
PPARA Q07869 2/20 0.34
CCR5 P51681 3/20 0.33
CYP2D6 P10635 1/20 0.33
GHSR Q92847 1/20 0.33
LRRK2 Q5S007 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19905836 0.95 JAK1 (0.37) JAK1JAK3JAK2IDO1KCNH2
SCHEMBL19905920 0.94 KDM4E (0.36) JAK1JAK3JAK2IDO1KCNH2
SCHEMBL19905832 0.89 MCHR1 (0.40) JAK1JAK3JAK2MCHR1KDM4E
SCHEMBL19905973 0.88 JAK2 (0.37) JAK1JAK3JAK2IDO1KCNH2
SCHEMBL19906238 0.86 KDM4E (0.35) IDO1KCNH2MCHR1KDM4EPTGDR2
SCHEMBL19906368 0.85 MCHR1 (0.43) MCHR1KDM4EPTGDR2MEN1ALDH1A1
SCHEMBL19906392 0.84 JAK1 (0.35) JAK1JAK3JAK2KDM4EPTGDR2
SCHEMBL19906223 0.84 MCHR1 (0.41) MCHR1CYP2D6
SCHEMBL19905942 0.83 DRD2 (0.40) KCNH2KDM4EPTGDR2MEN1ALDH1A1
SCHEMBL15332769 0.83 CYP3A4 (0.39) JAK1JAK3JAK2IDO1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed