SCHEMBL19906129

SCHEMBL19906129

Cc1cc2nc(-c3ccnc(-c4cnn(C)c4C)n3)sc2c(-c2ccc(Cl)cc2OC(C)(C)C)c1CC(=O)O

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EGFR P00533 4/20 0.33
SHMT1 P34896 2/20 0.33
SHMT2 P34897 2/20 0.33
IDH1 O75874 1/20 0.32
KDM4E B2RXH2 1/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
LMNA P02545 1/20 0.31
PTGS1 P23219 1/20 0.31
CYP2C19 P33261 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31
EIF4EBP1 Q13541 1/20 0.31
KDM2B Q8NHM5 1/20 0.30
KDM4C Q9H3R0 1/20 0.30
PPARD Q03181 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19906069 0.90 EGFR (0.35) EGFRSHMT1SHMT2IDH1KDM4E
SCHEMBL19906131 0.87 KDM4E (0.35) EGFRSHMT1SHMT2IDH1KDM4E
SCHEMBL19906087 0.86 KDM4E (0.32) SHMT1SHMT2KDM4ESMN1; SMN2LMNA
SCHEMBL19906150 0.86 RORC (0.33) SHMT1SHMT2KDM4EPTGS1CYP2C19
SCHEMBL19906391 0.85 KDM4E (0.33) KDM4ESMN1; SMN2LMNAPTGDR2PPARD
SCHEMBL19906374 0.83 POLQ (0.33) KDM4EPTGS1CYP2C19PTGDR2
SCHEMBL19906106 0.83 EIF4EBP1 (0.34) EIF4EBP1KDM2BKDM4CPPARD
SCHEMBL19906032 0.83 HRH4 (0.36) KDM4ELMNAEIF4EBP1PPARD
SCHEMBL19906017 0.82 KDM4E (0.32) KDM4ESMN1; SMN2LMNAPTGDR2EIF4EBP1
SCHEMBL19906161 0.82 KDM4E (0.35) SHMT1SHMT2KDM4ESMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed