SCHEMBL19906215

SCHEMBL19906215

Cc1cc2nc(-c3ccnc(-c4ccc5c(c4)OCC(=O)N5C)c3)sc2c(-c2ccc(Cl)cc2)c1CC(=O)OCC(C)(C)O

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
GABRG2 P18507 1/20 0.32
GABRB3 P28472 1/20 0.32
GABRA5 P31644 1/20 0.32
KDM1A O60341 2/20 0.31
PTGER3 P43115 1/20 0.31
IDH1 O75874 1/20 0.31
F10 P00742 1/20 0.30
USP2 O75604 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19906202 0.83 PTGER3 (0.40) PTGER3USP2HTT
SCHEMBL15342193 0.81 CYP11B1 (0.33) CYP11B1CYP11B2PTGER3IDH1F10
SCHEMBL15342601 0.81 CYP3A4 (0.35) CYP11B1CYP11B2PTGER3F10
SCHEMBL19906196 0.78 PTGER3 (0.34) PTGER3USP2HTT
SCHEMBL19906003 0.78 TRIM24 (0.41)
SCHEMBL19905990 0.77 GRM5 (0.39) CYP11B1CYP11B2PTGER3
SCHEMBL15342199 0.76 PTGER3 (0.35) PTGER3IDH1
SCHEMBL15342604 0.76 CYP3A4 (0.35) PTGER3
SCHEMBL19906264 0.76 PTGER3 (0.34) PTGER3IDH1
SCHEMBL19906330 0.76 KDM4E (0.33) HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed