SCHEMBL19906202

SCHEMBL19906202

Cc1cc2nc(-c3ccnc(-c4ccc5c(c4)N(C)C(=O)CO5)c3)sc2c(-c2ccc(Cl)cc2)c1CC(=O)O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGER3 P43115 1/20 0.40
KMO O15229 1/20 0.35
CPT1A P50416 1/20 0.35
CPT1B Q92523 1/20 0.35
APOBEC3A P31941 1/20 0.34
APOBEC3G Q9HC16 1/20 0.34
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
KLKB1 P03952 1/20 0.34
KDM4E B2RXH2 2/20 0.33
GPR55 Q9Y2T6 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
HTT P42858 2/20 0.33
TSHR P16473 1/20 0.33
USP2 O75604 1/20 0.32
HTR1A P08908 2/20 0.31
HTR1D P28221 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19906196 0.90 PTGER3 (0.34) PTGER3KMOCPT1ACPT1BAPOBEC3A
SCHEMBL19906111 0.88 PTGER3 (0.38) PTGER3CPT1ACPT1BKLKB1KDM4E
SCHEMBL19906003 0.87 TRIM24 (0.41) KDM4EMEN1ALDH1A1KMT2APTGDR2
SCHEMBL19906264 0.87 PTGER3 (0.34) PTGER3PDE3AKDM4EMEN1ALDH1A1
SCHEMBL19905989 0.84 NSD2 (0.38) ALDH1A1
SCHEMBL15342604 0.84 CYP3A4 (0.35) PTGER3PDE3BPDE3A
SCHEMBL19905990 0.83 GRM5 (0.39) PTGER3KDM4EMEN1ALDH1A1KMT2A
SCHEMBL19906215 0.83 CYP11B1 (0.33) PTGER3HTTUSP2
SCHEMBL19905979 0.83 KDM4E (0.33) PTGER3CPT1ACPT1BKDM4EMEN1
SCHEMBL15342199 0.83 PTGER3 (0.35) PTGER3APOBEC3AAPOBEC3GPDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed