SCHEMBL19906229

SCHEMBL19906229

COc1ncc(-c2cc(-c3nc4cc(C)c(CC(=O)O)c(-c5ccc(Cl)cc5OC(C)(C)C)c4s3)ccn2)cn1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EIF4E P06730 2/20 0.36
KDM4E B2RXH2 2/20 0.34
PTGDR2 Q9Y5Y4 3/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.33
CTSA P10619 8/20 0.32
LMNA P02545 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
PPARD Q03181 2/20 0.32
SHMT1 P34896 2/20 0.32
PTGS1 P23219 1/20 0.32
CYP2C19 P33261 1/20 0.32
CDC7 O00311 1/20 0.31
DBF4 Q9UBU7 1/20 0.31
SHMT2 P34897 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19906268 0.93 EIF4E (0.38) EIF4EKDM4EPTGDR2MEN1ALDH1A1
SCHEMBL19906137 0.91 PTGDR2 (0.39) EIF4EKDM4EPTGDR2MEN1ALDH1A1
SCHEMBL19906366 0.91 CTSA (0.34) KDM4EPTGDR2MEN1ALDH1A1KMT2A
SCHEMBL19906369 0.90 KDM4E (0.38) KDM4EPTGDR2MEN1ALDH1A1KMT2A
SCHEMBL19906060 0.90 KDM4E (0.38) EIF4EKDM4EPTGDR2MEN1ALDH1A1
SCHEMBL19905873 0.88 SHMT1 (0.32) KDM4EPTGDR2MEN1ALDH1A1KMT2A
SCHEMBL19906236 0.88 PTGDR2 (0.38) EIF4EKDM4EPTGDR2MEN1ALDH1A1
SCHEMBL19906291 0.87 PTGDR2 (0.33) EIF4EKDM4EPTGDR2MEN1ALDH1A1
SCHEMBL19906288 0.87 CSF1R (0.35) KDM4EPTGDR2MEN1ALDH1A1KMT2A
SCHEMBL19906328 0.87 PTGER1 (0.34) EIF4EKDM4EPTGDR2MEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed