SCHEMBL19906325

SCHEMBL19906325

COc1cc(-c2cccc(-c3nc4cc(C)c(CC(=O)O)c(-c5ccc(Cl)cc5)c4s3)c2)ccn1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.44
KDM4E B2RXH2 3/20 0.40
PTGDR2 Q9Y5Y4 9/20 0.39
KMT2A Q03164 3/20 0.39
ALDH1A1 P00352 2/20 0.39
MEN1 O00255 2/20 0.39
WNT3A P56704 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
HPGD P15428 1/20 0.38
CYP2C19 P33261 1/20 0.38
CYP19A1 P11511 1/20 0.36
SLC13A5 Q86YT5 1/20 0.35
MAPT P10636 1/20 0.35
LRRK2 Q5S007 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19906322 0.88 CNR1 (0.38) CNR1KDM4EPTGDR2KMT2AALDH1A1
SCHEMBL19906064 0.87 KDM4E (0.41) KDM4EPTGDR2KMT2AALDH1A1MEN1
SCHEMBL19905797 0.85 EIF4E (0.39) KDM4EPTGDR2KMT2AALDH1A1MEN1
SCHEMBL19906088 0.84 KDM4E (0.42) KDM4EPTGDR2KMT2AALDH1A1MEN1
SCHEMBL19905876 0.84 PTGDR2 (0.42) KDM4EPTGDR2KMT2AALDH1A1MEN1
SCHEMBL19905964 0.84 PTGDR2 (0.37) CNR1KDM4EPTGDR2KMT2AALDH1A1
SCHEMBL19906275 0.83 PTGDR2 (0.37) KDM4EPTGDR2KMT2AALDH1A1MEN1
SCHEMBL19906164 0.83 DYRK1A (0.40) KDM4EMAPT
SCHEMBL19906090 0.83 MEN1 (0.39) KDM4EPTGDR2KMT2AALDH1A1MEN1
SCHEMBL19906236 0.82 PTGDR2 (0.38) KDM4EPTGDR2KMT2AALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed