SCHEMBL19905964

SCHEMBL19905964

COc1ccc2ccc(-c3cc(-c4nc5cc(C)c(CC(=O)O)c(-c6ccc(Cl)cc6)c5s4)ccn3)cc2n1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 9/20 0.37
KDM4E B2RXH2 3/20 0.35
ALDH1A1 P00352 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CYP2C19 P33261 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
HPGD P15428 1/20 0.32
PTGS1 P23219 1/20 0.32
PPARD Q03181 2/20 0.32
MAP4K4 O95819 1/20 0.32
PTPN11 Q06124 1/20 0.31
CNR1 P21554 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19906275 0.94 PTGDR2 (0.37) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906291 0.89 PTGDR2 (0.33) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906249 0.88 ALDH1A1 (0.43) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906236 0.86 PTGDR2 (0.38) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906120 0.84 KDM4E (0.34) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906325 0.84 CNR1 (0.44) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906015 0.83 PIK3CG (0.38) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19905817 0.83 PTGDR2 (0.38) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906240 0.83 PTGDR2 (0.38) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19905802 0.83 MAP4K4 (0.43) PTGDR2KDM4EALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed