SCHEMBL19909299

SCHEMBL19909299

c1ccc(-c2cc3cc(-c4cccnn4)cnc3[nH]2)cc1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.51
PIK3CG P48736 1/20 0.46
KIT P10721 5/20 0.46
RIPK1 Q13546 7/20 0.45
CCNB2 O95067 3/20 0.43
CDK1 P06493 3/20 0.43
CCNB1 P14635 3/20 0.43
CCNB3 Q8WWL7 3/20 0.43
CDK5 Q00535 2/20 0.43
CDK5R1 Q15078 2/20 0.43
GSK3A P49840 1/20 0.43
GSK3B P49841 1/20 0.43
ULK1 O75385 2/20 0.42
ADORA2A P29274 1/20 0.42
ADORA1 P30542 1/20 0.42
NPY5R Q15761 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23912153 0.78 BRD4 (0.57) BRD4PIK3CGKITCCNB2CDK1
SCHEMBL19909156 0.78 BRD4 (0.51) BRD4PIK3CGKITRIPK1CCNB2
SCHEMBL18944010 0.78 BRD4 (0.51) BRD4PIK3CGKITRIPK1CCNB2
SCHEMBL18918667 0.75 ULK1 (0.59) BRD4PIK3CGKITULK1
SCHEMBL23912160 0.75 BRD4 (0.48) BRD4PIK3CGKITRIPK1CCNB2
SCHEMBL30236422 0.73 KIT (0.68) KIT
SCHEMBL15824723 0.73 KIT (0.68) KIT
SCHEMBL1778505 0.73 RIPK1 (0.74) RIPK1CCNB2CDK1CCNB1CCNB3
SCHEMBL15020472 0.72 CYP19A1 (0.54) BRD4PIK3CGKITRIPK1CCNB2
SCHEMBL1772615 0.72 RIPK1 (0.54) BRD4PIK3CGKITRIPK1CCNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2935248-B1 COMPOUNDS AND METHODS FOR KINASE MODULATION, AND INDICATIONS THEREFOR PLEXXIKON INC (US) 2018-02-28 EP disclosed