SCHEMBL19909508

SCHEMBL19909508

Cc1ccc(-c2ccc3c4ccc(-c5ccc(C#N)cc5)cc4n(-c4cc(C#N)cc(-n5c6cc(-c7ccc(C#N)cc7)ccc6c6ccc(-c7ccc(C#N)cc7)cc65)c4-c4ccncc4)c3c2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 2/20 0.42
FLT3 P36888 2/20 0.41
MAPKAPK2 P49137 1/20 0.40
ALDH1A1 P00352 1/20 0.37
CYP2A6 P11509 1/20 0.37
MAPK14 Q16539 2/20 0.36
CSNK1A1 P48729 1/20 0.36
CSNK1D P48730 1/20 0.36
CYP11B2 P19099 2/20 0.36
CYP11B1 P15538 1/20 0.36
BRAF P15056 1/20 0.35
KDR P35968 1/20 0.35
METAP2 P50579 1/20 0.35
PIK3CD O00329 1/20 0.35
PIK3CA P42336 1/20 0.35
PIK3CB P42338 1/20 0.35
MTOR P42345 1/20 0.35
PIK3CG P48736 1/20 0.35
KDM1A O60341 2/20 0.34
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19913161 0.98 FLT3 (0.40) CHEK1FLT3MAPKAPK2ALDH1A1MAPK14
SCHEMBL19919611 0.94 FLT3 (0.42) CHEK1FLT3MAPK14CSNK1A1CSNK1D
SCHEMBL19908939 0.92 MAPK14 (0.40) CHEK1FLT3MAPKAPK2ALDH1A1MAPK14
SCHEMBL19908940 0.89 GRM5 (0.39) CHEK1FLT3MAPK14CSNK1A1CSNK1D
SCHEMBL19913138 0.89 MAPK14 (0.36) FLT3ALDH1A1MAPK14CSNK1A1CSNK1D
SCHEMBL19909478 0.88 FLT3 (0.41) CHEK1FLT3MAPK14CSNK1A1CSNK1D
SCHEMBL19909067 0.88 MAPKAPK2 (0.39) CHEK1FLT3MAPKAPK2ALDH1A1CYP2A6
SCHEMBL19913158 0.87 MAPK14 (0.45) CHEK1FLT3ALDH1A1MAPK14CYP11B2
SCHEMBL25658975 0.87 PDE1C (0.41) CHEK1MAPKAPK2ALDH1A1CYP2A6KDM1A
SCHEMBL19913152 0.87 IMPDH2 (0.39) FLT3MAPK14CSNK1A1CSNK1DCYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3287451-A1 ORGANIC MOLECULES, IN PARTICULAR FOR USE IN ORGANIC OPTOELECTRONIC DEVICES CYNORA GMBH (DE) 2018-02-28 EP disclosed