SCHEMBL19909686

SCHEMBL19909686

NC(=O)c1sc(N2CCCC2)nc1-c1ccc(Oc2ccccc2)cc1

nearest known ligand 0.63

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.63
HTT P42858 3/20 0.63
NPSR1 Q6W5P4 2/20 0.63
BTK Q06187 12/20 0.62
SMN1; SMN2 Q16637 2/20 0.59
TDP1 Q9NUW8 2/20 0.59
ALOX5 P09917 2/20 0.59
MEN1 O00255 1/20 0.53
MAPT P10636 1/20 0.53
KMT2A Q03164 1/20 0.53
SCN9A Q15858 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19909712 0.99 ALDH1A1 (0.65) ALDH1A1HTTNPSR1BTKSMN1; SMN2
SCHEMBL16075347 0.90 BTK (0.56) ALDH1A1HTTNPSR1BTKSMN1; SMN2
SCHEMBL19909657 0.88 BTK (0.66) ALDH1A1HTTNPSR1BTKSMN1; SMN2
SCHEMBL16075279 0.86 BTK (0.66) BTK
SCHEMBL16075270 0.84 BTK (0.66) BTK
SCHEMBL16075328 0.84 BTK (0.50) ALDH1A1HTTNPSR1BTK
SCHEMBL19909740 0.84 BTK (0.50) ALDH1A1HTTNPSR1BTKSMN1; SMN2
SCHEMBL16075346 0.83 BTK (0.53) ALDH1A1HTTNPSR1BTKSCN9A
SCHEMBL19909753 0.83 ALDH1A1 (0.62) ALDH1A1HTTNPSR1SMN1; SMN2TDP1
SCHEMBL16075300 0.82 BTK (0.53) ALDH1A1HTTNPSR1BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970163-B1 5-THIAZOLECARBOXAMIDE DERVATIVES AND THEIR USE AS BTK INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2018-02-28 EP disclosed