SCHEMBL19909887

SCHEMBL19909887

CC1(C)CNC(c2cccc(F)c2)C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 3/20 0.44
RCOR1 Q9UKL0 1/20 0.44
L3MBTL1 Q9Y468 3/20 0.40
CA1 P00915 1/20 0.39
IDO1 P14902 1/20 0.38
CHRNA1 P02708 1/20 0.38
CHRNB1 P11230 1/20 0.38
CHRNB2 P17787 1/20 0.38
SLC6A2 P23975 1/20 0.38
CHRNB4 P30926 1/20 0.38
SLC6A4 P31645 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNA4 P43681 1/20 0.38
SLC6A3 Q01959 1/20 0.38
ALDH1A1 P00352 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
HTR2B P41595 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL455752 0.87 KDM1A (0.42) KDM1ARCOR1L3MBTL1CA1IDO1
SCHEMBL433347 0.83 KDM1A (0.41) KDM1ARCOR1L3MBTL1CA1IDO1
SCHEMBL430807 0.83 KDM1A (0.41) KDM1ARCOR1L3MBTL1CA1IDO1
SCHEMBL27881449 0.82 KDM1A (0.43) KDM1ARCOR1L3MBTL1CHRNA1CHRNB1
SCHEMBL8221834 0.82 KDM1A (0.43) KDM1ARCOR1IDO1CHRNA1CHRNB1
SCHEMBL3574526 0.80 KDM1A (0.44) KDM1AALDH1A1
SCHEMBL17724399 0.77 KDM1A (0.44) KDM1ARCOR1L3MBTL1CA1IDO1
SCHEMBL456182 0.75 KDM1A (0.40) KDM1ARCOR1L3MBTL1CA1CHRNA1
SCHEMBL20703377 0.74 KDM1A (0.39) KDM1ARCOR1L3MBTL1CA1IDO1
SCHEMBL14047341 0.73 QDPR (0.41) L3MBTL1ALDH1A1CYP3A4PKMTAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3106463-B1 SUBSTITUTED PYRAZOLO[1,5-]PYRIMIDINE COMPOUNDS AS TRK KINASE INHIBITORS ARRAY BIOPHARMA INC (US) 2018-02-28 EP disclosed