SCHEMBL19915958

SCHEMBL19915958

CCOc1c(C)cc2cncn2c1C(=O)OC

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.36
GAA P10253 3/20 0.36
MAPK1 P28482 2/20 0.36
IDO1 P14902 1/20 0.35
TBXAS1 P24557 1/20 0.35
ALDH1A1 P00352 3/20 0.33
ATM Q13315 2/20 0.33
HTT P42858 3/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
KDM4E B2RXH2 3/20 0.32
MAPT P10636 2/20 0.32
S1PR1 P21453 1/20 0.32
GLA P06280 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
ALOX15 P16050 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21060531 0.76 IDO1 (0.51) TSHRGAAMAPK1IDO1TBXAS1
SCHEMBL28701542 0.73 TBXAS1 (0.35) TSHRGAAMAPK1IDO1TBXAS1
SCHEMBL22445945 0.70 CYP3A4 (0.44) GAATBXAS1ALDH1A1SMN1; SMN2KDM4E
SCHEMBL19915935 0.70 IDO1 (0.39) TSHRGAAMAPK1IDO1TBXAS1
SCHEMBL28708782 0.70 ALDH1A1 (0.40) TSHRMAPK1IDO1TBXAS1ALDH1A1
SCHEMBL18137441 0.68 CYP2C9 (0.41) GAAMAPK1TBXAS1ALDH1A1HTT
SCHEMBL21113341 0.68 ALDH1A1 (0.39) TSHRGAATBXAS1ALDH1A1SMN1; SMN2
SCHEMBL19915857 0.67 IDO1 (0.39) TSHRGAAMAPK1IDO1TBXAS1
SCHEMBL28686852 0.67 KCNH2 (0.33) TSHRMAPK1IDO1TBXAS1ALDH1A1
SCHEMBL18137446 0.67 CYP2C9 (0.40) TSHRGAAMAPK1TBXAS1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3505517-A1 FUSED HETEROCYCLIC DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF Beijing InnoCare Pharma Tech Co., Ltd. (CN) 2019-07-03 EP disclosed
WO-2018036414-A1 FUSED HETEROCYCLIC DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 北京诺诚健华医药科技有限公司 2018-03-01 WO disclosed