SCHEMBL19917016

SCHEMBL19917016

Cc1nc(N)c2nnn(C)c2n1

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 4/20 0.44
ADORA2A P29274 3/20 0.44
PDE8B O95263 9/20 0.43
PDE8A O60658 2/20 0.33
ADORA2B P29275 1/20 0.33
ADORA3 P0DMS8 1/20 0.30
CDK1 P06493 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13347013 0.82 CDK1 (0.41) ADORA2APDE8BADORA3CDK1
SCHEMBL10307719 0.79 CA12 (0.33)
SCHEMBL21159333 0.78 PDE8B (0.43) ADORA1ADORA2APDE8BPDE8AADORA2B
SCHEMBL14134555 0.76 PDE8B (0.43) ADORA1ADORA2APDE8BPDE8AADORA2B
SCHEMBL26533052 0.76 PDE8B (0.41) ADORA1ADORA2APDE8BPDE8AADORA2B
SCHEMBL21138202 0.76 PDE8B (0.41) ADORA1ADORA2APDE8BPDE8AADORA2B
SCHEMBL13788521 0.71 TP53 (0.30)
SCHEMBL21138214 0.70 PDE8B (0.51) ADORA1ADORA2APDE8BADORA3
SCHEMBL21183232 0.69 DYRK1A (0.38) ADORA1ADORA2A
SCHEMBL13335021 0.69 ADORA1 (0.57) ADORA1ADORA2APDE8BADORA2BADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018038265-A1 BICYCLIC NITROGENATED HETEROCYCLIC COMPOUND 田辺三菱製薬株式会社 2018-03-01 WO disclosed