SCHEMBL1992184

SCHEMBL1992184

OC(c1ccncc1)c1c[nH]c2ccccc12

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.61
HSD17B10 Q99714 2/20 0.50
IMPDH2 P12268 1/20 0.50
MAPK1 P28482 1/20 0.50
AHR P35869 2/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
GPR84 Q9NQS5 3/20 0.47
FFAR1 O14842 2/20 0.47
HTR2A P28223 1/20 0.44
HTR2C P28335 1/20 0.44
HTR2B P41595 1/20 0.44
NOD2 Q9HC29 1/20 0.44
MGAM O43451 1/20 0.43
GAA P10253 1/20 0.43
SI P14410 1/20 0.43
MGAM2 Q2M2H8 1/20 0.43
SRC P12931 1/20 0.42
KIF20A O95235 1/20 0.42
CYP2D6 P10635 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13763231 0.86 MAPT (0.59) MAPTMAPK1AHRMEN1KMT2A
SCHEMBL7290548 0.83 MAPT (0.59) MAPTHSD17B10IMPDH2MAPK1AHR
SCHEMBL30913604 0.83 MAPT (0.59) MAPTHSD17B10IMPDH2MAPK1AHR
SCHEMBL8213938 0.82 MAPT (0.67) MAPTHSD17B10AHRMEN1KMT2A
SCHEMBL4266740 0.81 MAPT (0.48) MAPTAHRGPR84NOD2MGAM
SCHEMBL28767073 0.81 MAPT (0.54) MAPTAHRMEN1KMT2AGPR84
SCHEMBL18364667 0.81 MAPT (0.54) MAPTAHRMEN1KMT2AGPR84
SCHEMBL27714368 0.81 MEN1 (0.56) MAPTHSD17B10MAPK1AHRMEN1
SCHEMBL13763230 0.81 MGAM (0.58) MAPTMAPK1AHRMEN1KMT2A
SCHEMBL27714156 0.81 MAPT (0.54) MAPTHSD17B10AHRMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011079105-A1 NOVEL THIENOPYRROLE COMPOUNDS ABBOTT LABORATORIES (US) 2011-06-30 WO disclosed
WO-2011079105-A1 NOVEL THIENOPYRROLE COMPOUNDS ABBOTT LABORATORIES (US) 2011-06-30 WO disclosed
US-20110152243-A1 NOVEL THIENOPYRROLE COMPOUNDS ABBOTT LABORATORIES (US) 2011-06-23 US disclosed
US-20110152243-A1 NOVEL THIENOPYRROLE COMPOUNDS ABBOTT LABORATORIES (US) 2011-06-23 US disclosed
US-20110152243-A1 NOVEL THIENOPYRROLE COMPOUNDS ABBOTT LABORATORIES (US) 2011-06-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110152243-A1 NOVEL THIENOPYRROLE COMPOUNDS TPMT, TSLP, THPO MAPT 3071/4885HSD17B10 2995/4885IMPDH2 359/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.