SCHEMBL19935331

SCHEMBL19935331

CCCCN(C)OC(=O)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 0.50
L3MBTL1 Q9Y468 1/20 0.46
CES2 O00748 3/20 0.45
CES1 P23141 3/20 0.45
TDP1 Q9NUW8 1/20 0.44
CYP1A2 P05177 3/20 0.44
GAA P10253 2/20 0.44
CYP2D6 P10635 2/20 0.44
HPGD P15428 1/20 0.44
CYP2C19 P33261 1/20 0.44
TSHR P16473 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
DRD3 P35462 2/20 0.43
SCN1A P35498 2/20 0.43
SLC6A3 Q01959 2/20 0.43
KCNH2 Q12809 2/20 0.43
SCN2A Q99250 2/20 0.43
SCN3A Q9NY46 2/20 0.43
MAOA P21397 1/20 0.43
CNR1 P21554 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5678485 0.90 LMNA (0.53) LMNACES2CES1TDP1CYP1A2
SCHEMBL28920596 0.85 TDP1 (0.43) LMNATDP1CYP1A2CYP2D6CYP2C19
SCHEMBL11850307 0.85 LMNA (0.51) LMNAL3MBTL1CES2CES1TDP1
SCHEMBL27267377 0.83 TDP1 (0.41) LMNATDP1CYP1A2CYP2D6HPGD
SCHEMBL4050408 0.82 LMNA (0.52) LMNATDP1CYP1A2CYP2D6HPGD
SCHEMBL11530129 0.82 LMNA (0.49) LMNAL3MBTL1CES2CES1TDP1
SCHEMBL26179405 0.81 TSHR (0.46) LMNATDP1CYP1A2CYP2D6HPGD
Hydrochloric Acid SCHEMBL9134016 0.80 LMNA (0.44) LMNAL3MBTL1CES2CES1TDP1
SCHEMBL21673638 0.80 TSHR (0.48) LMNATDP1CYP1A2CYP2D6HPGD
SCHEMBL27851129 0.80 LMNA (0.50) LMNAL3MBTL1CES2CES1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3848372-A1 FUSED TRICYCLIC PYRIDAZINONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS Novartis AG (CH) 2021-07-14 EP disclosed
EP-3504214-B1 FUSED TRICYCLIC PYRIDAZINONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2020-12-02 EP disclosed
WO-2018042303-A1 FUSED TRICYCLIC PYRIDAZINONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2018-03-08 WO disclosed